SCHEMBL7470368

SCHEMBL7470368

Cc1nc(S(=O)(=O)N2CCC[C@H]2C(=O)N[C@@H](Cc2ccc(O)cc2)C(=O)OC(C)(C)C)c[nH]1

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 4/20 0.43
ITGB1 P05556 7/20 0.41
CACNA1B Q00975 6/20 0.41
LY96 Q9Y6Y9 1/20 0.41
ITGB7 P26010 1/20 0.41
ITGA5 P08648 3/20 0.41
ITGAV P06756 2/20 0.38
ITGA2 P17301 1/20 0.38
GAA P10253 1/20 0.38
MEN1 O00255 1/20 0.37
POLB P06746 1/20 0.37
MAPT P10636 1/20 0.37
MAPK1 P28482 1/20 0.37
KMT2A Q03164 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
GPR55 Q9Y2T6 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7390739 0.90 ITGA4 (0.43) ITGA4ITGB1ITGB7ITGA5ITGAV
SCHEMBL5608873 0.89 ITGB1 (0.44) ITGA4ITGB1CACNA1BITGB7ITGA5
SCHEMBL7408832 0.84 ITGB1 (0.47) ITGA4ITGB1ITGB7ITGA5ITGA2
SCHEMBL6429310 0.84 ITGB1 (0.51) ITGA4ITGB1ITGB7ITGA5ITGAV
SCHEMBL6712483 0.83 ITGA4 (0.57) ITGA4ITGB1ITGA5ITGAVGAA
SCHEMBL6714478 0.83 ITGA4 (0.43) ITGA4ITGB1CACNA1BLY96ITGA5
SCHEMBL3850851 0.83 ALDH1A1 (0.43) ITGA4ITGB1CACNA1BITGB7GAA
SCHEMBL6709349 0.81 ITGA4 (0.49) ITGA4ITGB1ITGA5ITGAVGAA
SCHEMBL6714722 0.81 ITGA4 (0.47) ITGA4ITGB1CACNA1BITGB7ITGA5
SCHEMBL6367710 0.80 ITGB1 (0.57) ITGA4ITGB1ITGB7ITGA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0994896-A1 SULFONYLATED DIPEPTIDE COMPOUNDS WHICH INHIBIT LEUKOCYTE ADHESION MEDIATED BY VLA-4 Elan Pharmaceuticals, Inc. (US) 2000-04-26 EP disclosed
WO-1999006437-A1 SULFONYLATED DIPEPTIDE COMPOUNDS WHICH INHIBIT LEUKOCYTE ADHESION MEDIATED BY VLA-4 ELAN PHARMACEUTICALS INC. (US) 1999-02-11 WO disclosed