SCHEMBL7470554

SCHEMBL7470554

O=[N+]([O-])c1ccc(N(CCO)CCO)c(C(F)(F)F)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 12/20 0.53
POLB P06746 2/20 0.43
PDE7A Q13946 1/20 0.42
HTT P42858 4/20 0.42
TP53 P04637 1/20 0.42
MAPT P10636 5/20 0.41
MEN1 O00255 5/20 0.41
KMT2A Q03164 5/20 0.41
LMNA P02545 4/20 0.41
PKM P14618 2/20 0.41
MAPK1 P28482 1/20 0.41
GAA P10253 2/20 0.40
NSD2 O96028 1/20 0.40
NCOA1 Q15788 1/20 0.40
NCOA3 Q9Y6Q9 1/20 0.40
TSHR P16473 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
AR P10275 3/20 0.39
AKR1C3 P42330 1/20 0.39
AKR1C2 P52895 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7478286 0.87 ALDH1A1 (0.45) ALDH1A1POLBPDE7AHTTTP53
SCHEMBL2088798 0.81 ALDH1A1 (0.51) ALDH1A1POLBHTTTP53MAPT
SCHEMBL110420 0.79 ALDH1A1 (0.52) ALDH1A1POLBHTTTP53MAPT
SCHEMBL7809597 0.79 ALDH1A1 (0.52) ALDH1A1POLBHTTTP53MAPT
SCHEMBL1984158 0.78 HSD17B10 (0.51) ALDH1A1POLBPDE7AHTTTP53
SCHEMBL7472206 0.78 ALDH1A1 (0.55) ALDH1A1POLBPDE7AHTTTP53
SCHEMBL186720 0.77 ALDH1A1 (0.55) ALDH1A1POLBPDE7AHTTTP53
SCHEMBL1408560 0.77 ALDH1A1 (0.48) ALDH1A1POLBPDE7AHTTTP53
SCHEMBL5923594 0.77 HTT (0.48) ALDH1A1POLBPDE7AHTTTP53
SCHEMBL15688012 0.76 ALDH1A1 (0.49) ALDH1A1POLBPDE7AHTTMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0711768-B1 BENZIMIDAZOLE DERIVATIVE MITSUI CHEMICALS INC (JP) 2002-02-13 EP disclosed
US-5852011-A Benzimidazole derivatives MITSUI CHEMICALS, INC. (JP) 1998-12-22 US disclosed
EP-0711768-A1 BENZIMIDAZOLE DERIVATIVE MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-05-15 EP disclosed