SCHEMBL7470577

SCHEMBL7470577

O=C(O)CN(Cc1ccccc1)[C@H]1CC[C@H](N2CCN(c3ccc4c(c3)CCNCC4)C2=O)CC1

nearest known ligand 0.43

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KHK P50053 6/20 0.43
F10 P00742 6/20 0.41
F2 P00734 5/20 0.41
HTR6 P50406 6/20 0.40
ACHE P22303 1/20 0.40
PRSS1 P07477 2/20 0.37
HTR2C P28335 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7470587 1.00 KHK (0.43) KHKF10F2HTR6ACHE
SCHEMBL7476660 0.85 KHK (0.42) KHKF10F2HTR6ACHE
SCHEMBL7476656 0.85 KHK (0.42) KHKF10F2HTR6ACHE
SCHEMBL7466178 0.79 KHK (0.43) KHKF10F2HTR6ACHE
SCHEMBL7466183 0.79 KHK (0.43) KHKF10F2HTR6ACHE
SCHEMBL7471860 0.78 ACHE (0.46) KHKF10F2HTR6ACHE
SCHEMBL7471852 0.78 ACHE (0.46) KHKF10F2HTR6ACHE
Hydrochloric Acid SCHEMBL8561905 0.77 KHK (0.41) KHKF10F2HTR6ACHE
Hydrochloric Acid SCHEMBL8558247 0.77 ACHE (0.46) KHKF10F2HTR6ACHE
Hydrochloric Acid SCHEMBL7422325 0.77 F10 (0.43) KHKF10F2HTR6ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0777667-A1 CYCLIC BENZAZEPINE UREA DERIVATIVES WITH AGGREGATION-INHIBITING EFFECT Dr. Karl Thomae GmbH (DE) 1997-06-11 EP disclosed
WO-1996005194-A1 CYCLIC BENZAZEPINE UREA DERIVATIVES WITH AGGREGATION-INHIBITING EFFECT DR. KARL THOMAE GMBH (DE) 1996-02-22 WO disclosed