SCHEMBL7466178

SCHEMBL7466178

O=C(O)CN[C@H]1CC[C@H](N2CCN(c3ccc4c(c3)CCNCC4)C2=O)CC1

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KHK P50053 6/20 0.43
HTR6 P50406 8/20 0.40
F2 P00734 1/20 0.38
F10 P00742 1/20 0.38
ITGB3 P05106 1/20 0.36
ITGA2B P08514 1/20 0.36
ACHE P22303 1/20 0.36
CYP17A1 P05093 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7466183 1.00 KHK (0.43) KHKHTR6F2F10ITGB3
SCHEMBL7465375 0.89 F10 (0.38) KHKF2F10ITGB3ITGA2B
SCHEMBL7465369 0.89 F10 (0.38) KHKF2F10ITGB3ITGA2B
Hydrochloric Acid SCHEMBL7468277 0.86 KHK (0.41) KHKHTR6F2F10
SCHEMBL7471860 0.83 ACHE (0.46) KHKHTR6F2F10ACHE
SCHEMBL7471852 0.83 ACHE (0.46) KHKHTR6F2F10ACHE
Hydrochloric Acid SCHEMBL8558247 0.82 ACHE (0.46) KHKHTR6F2F10ACHE
Hydrochloric Acid SCHEMBL8561905 0.82 KHK (0.41) KHKHTR6F2F10ITGB3
Hydrochloric Acid SCHEMBL7422325 0.82 F10 (0.43) KHKHTR6F2F10ITGB3
SCHEMBL7418636 0.81 MCHR1 (0.44) KHKHTR6F2F10ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0777667-A1 CYCLIC BENZAZEPINE UREA DERIVATIVES WITH AGGREGATION-INHIBITING EFFECT Dr. Karl Thomae GmbH (DE) 1997-06-11 EP claimed
WO-1996005194-A1 CYCLIC BENZAZEPINE UREA DERIVATIVES WITH AGGREGATION-INHIBITING EFFECT DR. KARL THOMAE GMBH (DE) 1996-02-22 WO claimed
EP-0777667-A1 CYCLIC BENZAZEPINE UREA DERIVATIVES WITH AGGREGATION-INHIBITING EFFECT Dr. Karl Thomae GmbH (DE) 1997-06-11 EP disclosed
WO-1996005194-A1 CYCLIC BENZAZEPINE UREA DERIVATIVES WITH AGGREGATION-INHIBITING EFFECT DR. KARL THOMAE GMBH (DE) 1996-02-22 WO disclosed