SCHEMBL7471880

SCHEMBL7471880

CCOC(=O)C1=C(CSCC2CO2)NC(C)=C(C(=O)OC)C1c1cccc(Cl)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 2/20 0.51
HIF1A Q16665 5/20 0.50
CYP2C9 P11712 5/20 0.50
MEN1 O00255 4/20 0.50
CYP1A2 P05177 4/20 0.50
CYP3A4 P08684 4/20 0.50
CYP2C19 P33261 4/20 0.50
KMT2A Q03164 4/20 0.50
MAPT P10636 3/20 0.50
POLB P06746 2/20 0.50
LMNA P02545 2/20 0.50
CYP2D6 P10635 2/20 0.50
TSHR P16473 2/20 0.50
NFKB1 P19838 2/20 0.50
THPO P40225 2/20 0.50
MAPK1 P28482 1/20 0.50
GPR55 Q9Y2T6 1/20 0.50
CACNA1B Q00975 5/20 0.47
KDM4E B2RXH2 2/20 0.46
HSD17B10 Q99714 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9808332 0.96 ABCC1 (0.48) ADORA3HIF1ACYP2C9MEN1CYP1A2
SCHEMBL9501260 0.90 ADORA3 (0.57) ADORA3HIF1ACYP2C9MEN1CYP1A2
SCHEMBL7419122 0.86 ADORA3 (0.53) ADORA3HIF1ACYP2C9MEN1CYP1A2
SCHEMBL7475640 0.86 HIF1A (0.71) ADORA3HIF1ACYP2C9MEN1CYP1A2
SCHEMBL7565092 0.85 ABCC1 (0.64) ADORA3MAPTLMNATSHRKDM4E
SCHEMBL9669318 0.83 ADORA3 (0.50) ADORA3HIF1ACYP2C9MEN1CYP1A2
SCHEMBL7318265 0.83 CACNA1B (0.51) ADORA3HIF1ACYP2C9MEN1CYP1A2
SCHEMBL9502243 0.83 ADORA3 (0.73) ADORA3HIF1ACYP2C9MEN1CYP1A2
SCHEMBL7423918 0.82 CACNA1F (0.69) ADORA3HIF1ACYP2C9MEN1CYP1A2
SCHEMBL7316147 0.82 ADORA3 (0.53) ADORA3HIF1ACYP2C9MEN1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5021436-A Antiulcer, anticoagulant, antiischaemic agent BOEHRINGER MANNHEIM ITALIA, S.P.A. (IT) 1991-06-04 US disclosed
US-4999362-A Hypotensive, Antiulcer, Cytoprotective, Antithrombotic Agents BOEHRINGER BIOCHEMIA ROBIN S.P.A. (IT) 1991-03-12 US disclosed
EP-0233228-A1 PHARMACEUTICALLY ACTIVE 2-THIOMETHYL-SUBSTITUTED-1,4-DIHYDROPYRIDINES BOEHRINGER MANNHEIM ITALIA S.P.A. (IT) 1987-08-26 EP disclosed
WO-1987000836-A1 PHARMACEUTICALLY ACTIVE 2-THIOMETHYL-SUBSTITUTED-1,4-DIHYDROPYRIDINES BOEHRINGER BIOCHEMIA ROBIN S.P.A. (IT) 1987-02-12 WO disclosed