SCHEMBL7472597

SCHEMBL7472597

COC(=O)C(=NO)C1=Nc2cc(Cl)ccc2C(c2ccccc2F)=NC1

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.42
CHRM1 P11229 1/20 0.40
AURKA O14965 2/20 0.40
TP53 P04637 1/20 0.40
SLC22A1 O15245 1/20 0.39
ABCB11 O95342 1/20 0.39
CYP3A4 P08684 1/20 0.39
DRD3 P35462 1/20 0.39
OPRK1 P41145 1/20 0.39
PDE4D Q08499 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7472591 1.00 LMNA (0.42) LMNACHRM1AURKATP53SLC22A1
SCHEMBL7313894 0.92 LMNA (0.44) LMNACHRM1AURKATP53SLC22A1
SCHEMBL7307232 0.92 LMNA (0.44) LMNACHRM1AURKATP53SLC22A1
SCHEMBL7473846 0.88 LMNA (0.45) LMNACHRM1AURKASLC22A1ABCB11
SCHEMBL7473843 0.88 LMNA (0.45) LMNACHRM1AURKASLC22A1ABCB11
SCHEMBL11371119 0.82 LMNA (0.42) LMNACHRM1AURKATP53SLC22A1
SCHEMBL11371073 0.82 LMNA (0.42) LMNACHRM1TP53SLC22A1ABCB11
SCHEMBL11366439 0.82 LMNA (0.42) LMNACHRM1TP53SLC22A1ABCB11
SCHEMBL11371076 0.82 LMNA (0.42) LMNACHRM1TP53SLC22A1ABCB11
SCHEMBL11366435 0.82 LMNA (0.42) LMNACHRM1TP53SLC22A1ABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1105392-B1 PROCESS FOR THE PREPARATION OF IMIDAZODIAZEPINE INTERMEDIATES ABBOTT LAB (US) 2002-09-04 EP disclosed
EP-1199308-A2 Process for the preparation of imidazodiazepine intermediates Abbott Laboratories (US) 2002-04-24 EP disclosed
US-20010014738-A1 PROCESS FOR THE PREPARATION OF IMIDAZODIAZEPINE INTERMEDIATES ABBOTT LABORATORIES 2001-08-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20010014738-A1 PROCESS FOR THE PREPARATION OF IMIDAZODIAZEPINE INTERMEDIATES CYP3A4, CYP4B1, CYP4A11 LMNA 1461/4885CHRM1 512/4885AURKA 569/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.