SCHEMBL7474024

SCHEMBL7474024

CCOC(=O)CN(C=C(C(=O)OCC)C(=O)OCC)Cc1ccccc1.CCOC(=O)CNCc1ccccc1

nearest known ligand 0.58

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PPID Q08752 1/20 0.47
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
SMN1; SMN2 Q16637 3/20 0.43
LTA4H P09960 5/20 0.42
NR1H4 Q96RI1 1/20 0.41
ALDH1A1 P00352 3/20 0.41
MAPT P10636 2/20 0.39
GAA P10253 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
PIN1 Q13526 1/20 0.38
TP53 P04637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4046871 0.90 MEN1 (0.54) PPIDMEN1KMT2ALTA4HNR1H4
SCHEMBL75205 0.79 PPID (0.69) PPIDSMN1; SMN2LTA4HALDH1A1MAPT
Hydrochloric Acid SCHEMBL3926946 0.78 PPID (0.68) PPIDSMN1; SMN2LTA4HALDH1A1MAPT
SCHEMBL2834704 0.77 ALDH1A1 (0.48) PPIDMEN1KMT2ASMN1; SMN2LTA4H
SCHEMBL4046878 0.74 TP53 (0.40) PPIDMEN1KMT2ASMN1; SMN2LTA4H
SCHEMBL19796001 0.73 ALDH1A1 (0.42) PPIDMEN1KMT2ASMN1; SMN2LTA4H
SCHEMBL12559711 0.73 PPID (0.64) PPIDMEN1KMT2ASMN1; SMN2LTA4H
SCHEMBL12894961 0.72 PPID (0.58) PPIDMEN1KMT2ASMN1; SMN2LTA4H
SCHEMBL10861409 0.72 KMT2A (0.55) MEN1KMT2ASMN1; SMN2NR1H4ALDH1A1
SCHEMBL13898294 0.70 MEN1 (0.48) PPIDMEN1KMT2ASMN1; SMN2LTA4H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1183033-A4 PYRROLOTRIAZINE INHIBITORS OF KINASES BRISTOL MYERS SQUIBB CO (US) 2002-07-17 EP disclosed
EP-1183033-A1 PYRROLOTRIAZINE INHIBITORS OF KINASES BRISTOL-MYERS SQUIBB COMPANY (US) 2002-03-06 EP disclosed
WO-2000071129-A1 PYRROLOTRIAZINE INHIBITORS OF KINASES BRISTOL-MYERS SQUIBB COMPANY (US) 2000-11-30 WO disclosed