SCHEMBL7474064

SCHEMBL7474064

O=C(c1ccc(Cl)nc1)c1cccc(F)c1F

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAPRT Q6XQN6 1/20 0.49
CES2 O00748 1/20 0.47
BCHE P06276 1/20 0.47
CES1 P23141 1/20 0.47
KCNQ3 O43525 6/20 0.42
KCNQ2 O43526 6/20 0.42
KCNE1 P15382 6/20 0.42
KCNQ1 P51787 6/20 0.42
BACE1 P56817 1/20 0.42
GAA P10253 1/20 0.42
KMT2A Q03164 1/20 0.41
L3MBTL1 Q9Y468 2/20 0.40
ALDH1A1 P00352 2/20 0.40
TDP1 Q9NUW8 1/20 0.40
MDM4 O15151 1/20 0.40
TP53 P04637 1/20 0.40
MDM2 Q00987 1/20 0.40
ALOX15 P16050 1/20 0.40
GRM4 Q14833 1/20 0.39
KDR P35968 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7676637 0.80 KMT2A (0.39) NAPRTCES2BCHECES1KCNQ3
SCHEMBL7679465 0.80 KMT2A (0.39) NAPRTCES2BCHECES1KCNQ3
SCHEMBL7440808 0.76 NAPRT (0.72) NAPRTKCNQ3KCNQ2KCNE1KCNQ1
SCHEMBL10633441 0.76 KCNQ3 (0.49) NAPRTCES2CES1KCNQ3KCNQ2
SCHEMBL7514511 0.75 KCNQ3 (0.60) KCNQ3KCNQ2KCNE1KCNQ1BACE1
SCHEMBL3440833 0.74 CES2 (0.74) CES2BCHECES1GAAKMT2A
SCHEMBL16460479 0.74 KCNQ3 (0.62) NAPRTCES2CES1KCNQ3KCNQ2
SCHEMBL8175947 0.74 CES2 (0.57) CES2BCHECES1GAAKMT2A
SCHEMBL4467915 0.74 NPC1 (0.62) NAPRTKCNQ3KCNQ2KCNE1KCNQ1
SCHEMBL20709029 0.74 CES2 (0.57) CES2BCHECES1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1077701-A4 ANTI-VIRAL COMPOUNDS LILLY CO ELI (US) 2002-03-20 EP disclosed
US-6358971-B1 FOR INHIBITING THE GROWTH OF A PICORNAVIRUS ELI LILLY AND COMPANY 2002-03-19 US disclosed
EP-1077701-A1 ANTI-VIRAL COMPOUNDS ELI LILLY AND COMPANY (US) 2001-02-28 EP disclosed
WO-1999059587-A1 ANTI-VIRAL COMPOUNDS ELI LILLY AND COMPANY (US) 1999-11-25 WO disclosed