SCHEMBL7475587

SCHEMBL7475587

Cc1c[nH]c(C(N)=O)c1N

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CCNC P24863 7/20 0.42
CDK8 P49336 7/20 0.42
GDA Q9Y2T3 1/20 0.41
NOTUM Q6P988 2/20 0.38
PDPK1 O15530 1/20 0.36
ALDH1A1 P00352 2/20 0.33
SLC9A1 P19634 1/20 0.33
LMNA P02545 2/20 0.32
TSHR P16473 2/20 0.32
KDM4E B2RXH2 2/20 0.32
PAX8 Q06710 1/20 0.32
MMP9 P14780 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
ATAD2 Q6PL18 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27479238 0.83 NOTUM (0.47) CCNCCDK8NOTUMKDM4EATAD2
SCHEMBL20157257 0.80 CCNC (0.51) CCNCCDK8GDANOTUMPDPK1
SCHEMBL16883380 0.78 KDM4E (0.40) NOTUMALDH1A1LMNATSHRKDM4E
Alcohol SCHEMBL27460337 0.76 NOTUM (0.41) CCNCCDK8NOTUMKDM4E
SCHEMBL2576551 0.75 ALDH1A1 (0.47) ALDH1A1LMNATSHRKDM4ESMN1; SMN2
SCHEMBL7560908 0.74 CCNC (0.50) CCNCCDK8GDANOTUMPDPK1
SCHEMBL13790182 0.72 CCNC (0.42) CCNCCDK8GDAALDH1A1LMNA
SCHEMBL1801972 0.70 NOTUM (0.47) CCNCCDK8GDANOTUMALDH1A1
SCHEMBL7116182 0.67 CCNC (0.47) CCNCCDK8NOTUMALDH1A1KDM4E
SCHEMBL1082611 0.67 NOTUM (0.65) CCNCCDK8NOTUMALDH1A1SLC9A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1183033-A4 PYRROLOTRIAZINE INHIBITORS OF KINASES BRISTOL MYERS SQUIBB CO (US) 2002-07-17 EP disclosed
EP-1183033-A1 PYRROLOTRIAZINE INHIBITORS OF KINASES BRISTOL-MYERS SQUIBB COMPANY (US) 2002-03-06 EP disclosed
WO-2000071129-A1 PYRROLOTRIAZINE INHIBITORS OF KINASES BRISTOL-MYERS SQUIBB COMPANY (US) 2000-11-30 WO disclosed