SCHEMBL7475764

SCHEMBL7475764

CC(=O)Nc1cccc(Nc2nccc(-c3ccncc3)n2)c1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 8/20 0.71
JAK3 P52333 1/20 0.68
PLK1 P53350 1/20 0.68
ABL1 P00519 9/20 0.65
BCR P11274 8/20 0.65
SRC P12931 6/20 0.65
PRKCA P17252 4/20 0.65
PRKCD Q05655 3/20 0.65
HDAC1 Q13547 2/20 0.64
HDAC6 Q9UBN7 2/20 0.64
PDGFRB P09619 5/20 0.60
PDGFRA P16234 5/20 0.60
PRKD3 O94806 1/20 0.59
PRKCG P05129 1/20 0.59
PRKCB P05771 1/20 0.59
PRKCH P24723 1/20 0.59
PRKCI P41743 1/20 0.59
PRKCE Q02156 1/20 0.59
PRKCQ Q04759 1/20 0.59
PRKCZ Q05513 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4375283 0.89 JAK2 (0.86) JAK2JAK3PLK1ABL1BCR
SCHEMBL7468958 0.89 ABL1 (0.76) JAK2PLK1ABL1BCRSRC
SCHEMBL7470447 0.87 JAK2 (0.79) JAK2JAK3PLK1ABL1BCR
Cyclohexane SCHEMBL5776808 0.86 ABL1 (0.63) JAK2ABL1BCRSRCPRKCA
SCHEMBL4895446 0.86 ABL1 (0.63) JAK2ABL1BCRSRCPRKCA
SCHEMBL3123409 0.85 ABL1 (0.82) JAK2ABL1BCRSRCPRKCA
SCHEMBL4905181 0.84 ABL1 (0.83) JAK2ABL1BCRSRCPRKCA
SCHEMBL4733852 0.84 PLK1 (0.84) JAK2JAK3PLK1ABL1BCR
SCHEMBL4378752 0.83 JAK2 (1.00) JAK2JAK3PLK1ABL1BCR
SCHEMBL4736493 0.83 PLK1 (0.83) JAK2JAK3PLK1ABL1BCR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0233461-B2 4,5,6-Substituted-2-pyrimidinamines AMERICAN CYANAMID CO (US) 2002-05-29 EP disclosed