SCHEMBL7475853

SCHEMBL7475853

c1cncc(OCCOc2sccc2N2CCNCC2)c1

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 7/20 0.45
CHRNA4 P43681 7/20 0.45
HTR6 P50406 1/20 0.43
CHRNA3 P32297 2/20 0.40
CHRNA7 P36544 2/20 0.40
CHRNA1 P02708 1/20 0.40
CHRNG P07510 1/20 0.40
CHRNB1 P11230 1/20 0.40
CHRNB4 P30926 1/20 0.40
CHRND Q07001 1/20 0.40
HTR1A P08908 1/20 0.39
SLC6A2 P23975 1/20 0.39
SLC6A4 P31645 1/20 0.39
SLC6A3 Q01959 1/20 0.39
PDE3B Q13370 1/20 0.38
PDE3A Q14432 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4315261 0.75 CHRNB2 (0.46) CHRNB2CHRNA4CHRNA3CHRNA7CHRNA1
SCHEMBL4320113 0.75 CHRNB2 (0.48) CHRNB2CHRNA4CHRNA3CHRNA7CHRNA1
SCHEMBL15986145 0.73 CHRNB2 (0.54) CHRNB2CHRNA4CHRNA3CHRNA7CHRNA1
SCHEMBL4307776 0.71 TSHR (0.58) CHRNB2CHRNA4
SCHEMBL4315272 0.71 CHRNB2 (0.44) CHRNB2CHRNA4HTR6
SCHEMBL2640059 0.71 TSHR (0.47) CHRNB2CHRNA4CHRNA3CHRNA7HTR1A
SCHEMBL4325786 0.70 CHRNB2 (0.43) CHRNB2CHRNA4CHRNA3CHRNA7CHRNA1
SCHEMBL4308694 0.70 CHRNB2 (0.43) CHRNB2CHRNA4HTR1A
SCHEMBL5335460 0.69 HTR1A (0.71) CHRNB2CHRNA4HTR6HTR1ASLC6A2
SCHEMBL4321095 0.68 TSHR (0.46) CHRNB2CHRNA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1178973-A2 NOVEL COMPOUNDS, THEIR USE AND PREPARATION Pharmacia AB (SE) 2002-02-13 EP disclosed
WO-2000076984-A2 NOVEL COMPOUNDS, THEIR USE AND PREPARATION BIOVITRUM AB (SE) 2000-12-21 WO disclosed