SCHEMBL7476622

SCHEMBL7476622

COc1cccc2c1CN(Nc1ccccn1)C2

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 6/20 0.42
RAB9A P51151 6/20 0.42
SMN1; SMN2 Q16637 4/20 0.42
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
GAA P10253 3/20 0.42
TP53 P04637 2/20 0.42
ALDH1A1 P00352 3/20 0.41
ALOX12 P18054 2/20 0.41
KDM4E B2RXH2 1/20 0.41
PKM P14618 1/20 0.40
HTT P42858 1/20 0.39
KDR P35968 1/20 0.38
DRD2 P14416 2/20 0.38
DRD3 P35462 2/20 0.38
ADRA1A P35348 1/20 0.38
ROCK2 O75116 1/20 0.38
DRD1 P21728 1/20 0.38
DRD5 P21918 1/20 0.38
TIPARP Q7Z3E1 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7477800 0.82 ALDH1A1 (0.40) NPC1RAB9ASMN1; SMN2MEN1KMT2A
SCHEMBL7481791 0.81 ALDH1A1 (0.41) NPC1RAB9ASMN1; SMN2MEN1KMT2A
SCHEMBL7474257 0.80 MEN1 (0.44) NPC1RAB9ASMN1; SMN2MEN1KMT2A
Hydrochloric Acid SCHEMBL7484737 0.80 ALDH1A1 (0.40) NPC1RAB9ASMN1; SMN2MEN1KMT2A
SCHEMBL7480365 0.78 CYP19A1 (0.44) SMN1; SMN2ALDH1A1DRD2DRD3ROCK2
SCHEMBL7477791 0.78 NPC1 (0.42) NPC1RAB9ASMN1; SMN2MEN1KMT2A
SCHEMBL27510166 0.72 MEN1 (0.35) NPC1RAB9ASMN1; SMN2MEN1KMT2A
SCHEMBL7485418 0.71 GAA (0.36) NPC1RAB9ASMN1; SMN2MEN1KMT2A
SCHEMBL7480185 0.70 GRIN2D (0.51) KDM4EHTTDRD2DRD3ADRA1A
SCHEMBL7482069 0.68 NPC1 (0.36) NPC1RAB9ASMN1; SMN2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0950056-B1 N-(PYRIDINYLAMINO)ISOINDOLINES AND RELATED COMPOUNDS AVENTIS PHARMA INC (US) 2002-09-18 EP claimed
EP-0950056-A2 N-(PYRIDINYLAMINO)ISOINDOLINES AND RELATED COMPOUNDS HOECHST MARION ROUSSEL, INC. (US) 1999-10-20 EP claimed
WO-1998029407-A2 N-(PYRIDINYLAMINO)ISOINDOLINES FOR TREATING ALZHEIMER'S AND DEPRESSION HOECHST MARION ROUSSEL, INC. (US) 1998-07-09 WO claimed
EP-0950056-B1 N-(PYRIDINYLAMINO)ISOINDOLINES AND RELATED COMPOUNDS AVENTIS PHARMA INC (US) 2002-09-18 EP disclosed
US-6004977-A ANTIDEPRESSANTS, COGNITION ACTIVATORS, AND ALZHEIMER'S DISEASE TREATMENT HOECHST MARION ROUSSEL, INC. (US) 1999-12-21 US disclosed
EP-0950056-A2 N-(PYRIDINYLAMINO)ISOINDOLINES AND RELATED COMPOUNDS HOECHST MARION ROUSSEL, INC. (US) 1999-10-20 EP disclosed
WO-1998029407-A2 N-(PYRIDINYLAMINO)ISOINDOLINES FOR TREATING ALZHEIMER'S AND DEPRESSION HOECHST MARION ROUSSEL, INC. (US) 1998-07-09 WO disclosed