SCHEMBL7477791

SCHEMBL7477791

COC(=O)Nc1cccc2c1CN(Nc1ccccn1)C2

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 9/20 0.42
RAB9A P51151 9/20 0.42
SMN1; SMN2 Q16637 3/20 0.42
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
CDK4 P11802 1/20 0.40
CCND2 P30279 1/20 0.40
MAPT P10636 1/20 0.39
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
PKM P14618 2/20 0.38
TP53 P04637 2/20 0.38
GAA P10253 2/20 0.38
F2 P00734 1/20 0.38
KDR P35968 1/20 0.37
ALOX12 P18054 1/20 0.37
CDK5 Q00535 1/20 0.36
CDK5R1 Q15078 1/20 0.36
RXFP1 Q9HBX9 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7477800 0.79 ALDH1A1 (0.40) NPC1RAB9ASMN1; SMN2KDM4EALDH1A1
SCHEMBL7476622 0.78 NPC1 (0.42) NPC1RAB9ASMN1; SMN2KDM4EALDH1A1
SCHEMBL7480814 0.78 KMT2A (0.46) NPC1RAB9ASMN1; SMN2KDM4EALDH1A1
SCHEMBL7481791 0.78 ALDH1A1 (0.41) NPC1RAB9ASMN1; SMN2KDM4EALDH1A1
Hydrochloric Acid SCHEMBL7484737 0.76 ALDH1A1 (0.40) NPC1RAB9ASMN1; SMN2KDM4EALDH1A1
SCHEMBL7474257 0.74 MEN1 (0.44) NPC1RAB9ASMN1; SMN2KDM4EALDH1A1
SCHEMBL27510166 0.73 MEN1 (0.35) NPC1RAB9ASMN1; SMN2KDM4EALDH1A1
SCHEMBL7485418 0.73 GAA (0.36) NPC1RAB9ASMN1; SMN2KDM4EALDH1A1
SCHEMBL17266541 0.71 NPC1 (0.66) NPC1RAB9ASMN1; SMN2KDM4EALDH1A1
SCHEMBL29655221 0.71 NPC1 (0.66) NPC1RAB9ASMN1; SMN2KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0950056-B1 N-(PYRIDINYLAMINO)ISOINDOLINES AND RELATED COMPOUNDS AVENTIS PHARMA INC (US) 2002-09-18 EP claimed
EP-0950056-A2 N-(PYRIDINYLAMINO)ISOINDOLINES AND RELATED COMPOUNDS HOECHST MARION ROUSSEL, INC. (US) 1999-10-20 EP claimed
WO-1998029407-A2 N-(PYRIDINYLAMINO)ISOINDOLINES FOR TREATING ALZHEIMER'S AND DEPRESSION HOECHST MARION ROUSSEL, INC. (US) 1998-07-09 WO claimed
EP-0950056-B1 N-(PYRIDINYLAMINO)ISOINDOLINES AND RELATED COMPOUNDS AVENTIS PHARMA INC (US) 2002-09-18 EP disclosed
US-6004977-A ANTIDEPRESSANTS, COGNITION ACTIVATORS, AND ALZHEIMER'S DISEASE TREATMENT HOECHST MARION ROUSSEL, INC. (US) 1999-12-21 US disclosed