SCHEMBL7477277

SCHEMBL7477277

Cc1ccc2c(c1)OC=C(CCl)N(CCCCN1CCC(c3ncnc4ccccc34)CC1)C2=O

nearest known ligand 0.48

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 8/20 0.36
HTR1A P08908 7/20 0.36
HTR2A P28223 7/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7462543 0.84 PARP1 (0.37) HTR1A
SCHEMBL7477282 0.81 DRD2 (0.34) DRD2HTR1AHTR2A
SCHEMBL7477239 0.79 DRD2 (0.38) DRD2HTR1AHTR2A
SCHEMBL7473425 0.79 HTR1A (0.40) HTR1A
SCHEMBL7470711 0.78 KCNH2 (0.51) DRD2HTR1AHTR2A
SCHEMBL7463338 0.78 DRD4 (0.46) DRD2
SCHEMBL7470708 0.77 DRD4 (0.40) DRD2HTR1A
SCHEMBL7473722 0.75 HTR1A (0.39) DRD2HTR1AHTR2A
SCHEMBL7473410 0.75 DRD2 (0.36) DRD2HTR1AHTR2A
SCHEMBL7471767 0.75 HTR1A (0.39) DRD2HTR1AHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0755930-B1 BENZOXAZEPINE DERIVATIVES, SALTS THEREOF, AND DRUGS CONTAINING THE SAME SUNTORY LTD (JP) 2002-07-31 EP disclosed
US-6337397-B1 A BENZOXAZEPINE DERIVATIVE FOR TREATMENT OF ANXIETY NEUROSIS, PHOBIAS, OBSESSIVE-COMPULSIVE DISORDERS, SCHIZOPHRENIA, POST-CARDIAC TRAUMA STRESS DISORDERS, DEPRESSION DISORDERS, PSYCHOSOMATIC DISORDERS AND OTHER PSYCHONEUROTIC DISORDERS, SUNTORY LIMITED (JP) 2002-01-08 US disclosed
US-6187769-B1 Benzoxazepine derivatives and their salts and medicaments containing the same SUNTORY LIMITED (JP) 2001-02-13 US disclosed
EP-0755930-A1 BENZOXAZEPINE DERIVATIVES, SALTS THEREOF, AND DRUGS CONTAINING THE SAME SUNTORY LIMITED (JP) 1997-01-29 EP disclosed