SCHEMBL7477368

SCHEMBL7477368

CCC(CC1CCCO1)c1cc(O)c(C(c2ccc(C)s2)C2CC2)c(=O)o1

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.34
MAPT P10636 5/20 0.34
HPGD P15428 4/20 0.34
KDM4E B2RXH2 4/20 0.34
POLB P06746 3/20 0.34
KMT2A Q03164 3/20 0.34
PKM P14618 1/20 0.34
TP53 P04637 1/20 0.33
RAB9A P51151 2/20 0.32
GAA P10253 1/20 0.32
NPC1 O15118 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
THRB P10828 1/20 0.31
TSHR P16473 1/20 0.31
HTT P42858 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7443483 0.98 ALDH1A1 (0.33) ALDH1A1MAPTHPGDKDM4EPOLB
SCHEMBL7473213 0.89 ALDH1A1 (0.35) ALDH1A1MAPTHPGDKDM4EPOLB
SCHEMBL7447423 0.87 ALDH1A1 (0.34) ALDH1A1MAPTHPGDKDM4EPOLB
SCHEMBL7445667 0.86 ALDH1A1 (0.31) ALDH1A1HPGDKMT2A
SCHEMBL7447084 0.86
SCHEMBL7450139 0.85 HPGD (0.38) ALDH1A1MAPTHPGDKDM4EPOLB
SCHEMBL7449599 0.85
SCHEMBL7444011 0.84 HPGD (0.37) ALDH1A1MAPTHPGDKDM4EPOLB
SCHEMBL6174809 0.83 HPGD (0.42) ALDH1A1HPGDKDM4EPKMRAB9A
SCHEMBL7438155 0.82 CCR5 (0.30) ALDH1A1HPGDKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0668860-B1 PYRAN-2-ONES AND 5,6-DIHYDROPYRAN-2-ONES USEFUL FOR TREATING HIV AND OTHER RETROVIRUSES UPJOHN CO (US) 2002-09-11 EP claimed
WO-1994011361-A1 PYRAN-2-ONES AND 5,6-DIHYDROPYRAN-2-ONES USEFUL FOR TREATING HIV AND OTHER RETROVIRUSES THE UPJOHN COMPANY (US) 1994-05-26 WO claimed
EP-1203770-A1 Pyran-2-ones and 5,6-dihydropyran-2-ones useful for treating hyperplasia and other diseases PHARMACIA & UPJOHN COMPANY (US) 2002-05-08 EP disclosed