SCHEMBL7477705

SCHEMBL7477705

Nc1ccc2c(c1)nc1snc(-c3ccccc3)n12

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.49
KMT2A Q03164 3/20 0.42
TLR9 Q9NR96 2/20 0.42
ATM Q13315 1/20 0.42
KDM4E B2RXH2 10/20 0.41
NPC1 O15118 5/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
FGFR1 P11362 1/20 0.41
HTT P42858 3/20 0.40
MAPT P10636 4/20 0.38
HPGD P15428 4/20 0.38
GAA P10253 3/20 0.38
RAB9A P51151 3/20 0.38
GLA P06280 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
MEN1 O00255 2/20 0.38
GFER P55789 2/20 0.38
PKM P14618 2/20 0.38
RCE1 Q9Y256 1/20 0.38
STAT1 P42224 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7479179 0.90 KMT2A (0.43) ALDH1A1KMT2ATLR9ATMKDM4E
SCHEMBL7477004 0.82 KDM4E (0.51) ALDH1A1KMT2AKDM4ENPC1HTT
SCHEMBL2326728 0.74 ALDH1A1 (0.70) ALDH1A1KMT2ATLR9ATMKDM4E
SCHEMBL31474854 0.72 ALDH1A1 (0.64) ALDH1A1KMT2ATLR9ATMKDM4E
SCHEMBL3158636 0.72 ALDH1A1 (0.67) ALDH1A1KMT2ATLR9ATMKDM4E
SCHEMBL7479438 0.70 CSNK1A1 (0.40) ALDH1A1KMT2AKDM4ENPC1HTT
SCHEMBL11441705 0.70 ALDH1A1 (0.68) ALDH1A1KMT2AKDM4ENPC1L3MBTL1
SCHEMBL7480580 0.67 CSNK1A1 (0.39) ALDH1A1KDM4ENPC1HTTMAPT
SCHEMBL2329961 0.66 ALDH1A1 (0.58) ALDH1A1KMT2AL3MBTL1MAPTRAB9A
SCHEMBL614951 0.66 ALDH1A1 (1.00) ALDH1A1KMT2AKDM4ENPC1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0883622-B1 PROTON PUMP INHIBITOR APOTEX INC (CA) 2002-05-15 EP claimed
US-6093738-A IMIDAZO(1,2-D)-THIADIAZOLE COMPOUNDS; PEPTIC ULCER TREATMENT KARIMIAN KHASHAYAR (CA) 2000-07-25 US claimed
CN-1216527-A Method for scavenging mercaptan APOTEX INC (CA) 1999-05-12 CN claimed
EP-0883622-B1 PROTON PUMP INHIBITOR APOTEX INC (CA) 2002-05-15 EP disclosed