SCHEMBL7478147

SCHEMBL7478147

O=C1Cc2c(cccc2OCCNCc2ccccc2)N1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 4/20 1.00
DRD4 P21917 4/20 1.00
DRD3 P35462 4/20 1.00
HTR6 P50406 4/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7480072 0.89 DRD2 (0.80) DRD2DRD4DRD3HTR6
SCHEMBL7485710 0.86 DRD2 (0.76) DRD2DRD4DRD3HTR6
SCHEMBL21538147 0.81 DRD2 (0.69) DRD2DRD4DRD3HTR6
SCHEMBL7475432 0.81 DRD2 (0.68) DRD2DRD4DRD3
SCHEMBL7482710 0.81 DRD2 (0.67) DRD2DRD4DRD3
SCHEMBL5638400 0.80 DRD2 (0.67) DRD2DRD4DRD3
SCHEMBL7474193 0.80 DRD2 (0.67) DRD2DRD4DRD3
SCHEMBL7443236 0.78 DRD2 (0.63) DRD2DRD4DRD3
SCHEMBL9385747 0.78 DRD2 (0.63) DRD2DRD4DRD3
Hydrochloric Acid SCHEMBL7443683 0.77 DRD2 (0.62) DRD2DRD4DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0923551-B1 4-AMINOETHOXY INDOLONE DERIVATIVES AMERICAN HOME PROD (US) 2002-06-05 EP claimed
US-5817690-A ANTIDOPAMINE AGENTS AMERICAN HOME PRODUCTS CORPORATION (US) 1998-10-06 US claimed
EP-0923551-B1 4-AMINOETHOXY INDOLONE DERIVATIVES AMERICAN HOME PROD (US) 2002-06-05 EP disclosed
EP-0923551-A1 4-AMINOETHOXY INDOLONE DERIVATIVES AMERICAN HOME PRODUCTS CORPORATION (US) 1999-06-23 EP disclosed
US-5817690-A ANTIDOPAMINE AGENTS AMERICAN HOME PRODUCTS CORPORATION (US) 1998-10-06 US disclosed
WO-1998008819-A1 4-AMINOETHOXY INDOLONE DERIVATIVES AMERICAN HOME PRODUCTS CORPORATION (US) 1998-03-05 WO disclosed