SCHEMBL7478259

SCHEMBL7478259

COC(=O)c1c(C(=O)OC(C)(C)C)cc2[nH]c(C)nc2c1O

nearest known ligand 0.38

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 12/20 0.38
CACNA1H O95180 1/20 0.34
CACNA1B Q00975 1/20 0.34
CACNA1C Q13936 1/20 0.34
PARP1 P09874 1/20 0.34
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7478263 0.81 MEN1 (0.33) NPSR1
SCHEMBL6583292 0.74 KCNH2 (0.42) DHODHPARP1
SCHEMBL6585161 0.72 PARP1 (0.46) DHODHPARP1
SCHEMBL6583248 0.71 DHODH (0.34) DHODHPARP1
SCHEMBL7333705 0.71 PARP1 (0.62) DHODHPARP1
SCHEMBL7421982 0.71 PARP1 (0.47) DHODHPARP1
SCHEMBL29893736 0.70 DHODH (0.38) DHODHPARP1CYP2C9CYP2C19NPSR1
SCHEMBL31177973 0.70 DHODH (0.38) DHODHPARP1CYP2C9CYP2C19NPSR1
SCHEMBL30938989 0.68 DYRK1A (0.40) DHODHPARP1
SCHEMBL8953009 0.68 PARP1 (0.47) DHODHPARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0865281-A4 NAPHTHYL-SUBSTITUTED BENZIMIDAZOLE DERIVATIVES AS ANTICOAGULANTS BERLEX LAB (US) 1999-07-28 EP disclosed
EP-0865281-A1 NAPHTHYL-SUBSTITUTED BENZIMIDAZOLE DERIVATIVES AS ANTICOAGULANTS BERLEX LABORATORIES, INC. (US) 1998-09-23 EP disclosed
WO-1997021437-A1 NAPHTHYL-SUBSTITUTED BENZIMIDAZOLE DERIVATIVES AS ANTICOAGULANTS BERLEX LABORATORIES, INC. (DE) 1997-06-19 WO disclosed