SCHEMBL6583248

SCHEMBL6583248

Cc1nc2c(C)c(N=C=S)c(C(=O)OC(C)(C)C)cc2[nH]1

nearest known ligand 0.36

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 11/20 0.34
PARP1 P09874 1/20 0.33
GABRA1 P14867 3/20 0.32
GABRG2 P18507 3/20 0.32
GABRB3 P28472 3/20 0.32
GABRA3 P34903 3/20 0.32
GABRA2 P47869 3/20 0.32
GABRA5 P31644 1/20 0.32
GABRA4 P48169 1/20 0.32
GABRA6 Q16445 1/20 0.32
HTT P42858 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6583253 0.85 GABRA1 (0.30) GABRA1GABRG2GABRB3GABRA3GABRA2
SCHEMBL6583292 0.75 KCNH2 (0.42) DHODHPARP1
SCHEMBL6585161 0.73 PARP1 (0.46) DHODHPARP1GABRA1GABRG2GABRB3
SCHEMBL7478259 0.71 DHODH (0.38) DHODHPARP1
SCHEMBL7333705 0.70 PARP1 (0.62) DHODHPARP1
SCHEMBL6954591 0.65 GABRA1 (0.30) GABRA1GABRG2GABRB3GABRA3GABRA2
SCHEMBL6954595 0.65 GABRA1 (0.30) GABRA1GABRG2GABRB3GABRA3GABRA2
SCHEMBL8132021 0.63 DHODH (0.54) DHODHPARP1
SCHEMBL5822166 0.62 ALDH1A1 (0.42) GABRA1GABRG2GABRB3GABRA3GABRA2
SCHEMBL6585164 0.62 HSP90AA1 (0.36) GABRA1GABRG2GABRB3GABRA3GABRA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1037887-B1 5-(2-IMIDAZOLINYLAMINO)-BENZIMIDAZOLE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS .ALPHA.-ADRENOCEPTOR AGONISTS WITH IMPROVED METABOLIC STABILITY PROCTER & GAMBLE (US) 2004-07-14 EP disclosed