SCHEMBL747836

SCHEMBL747836

O=C(N1CCCCCC1)N1CCC2(CC1)CCN(c1ccc(OC(F)(F)F)cc1)C2

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 12/20 0.49
ITGB3 P05106 6/20 0.47
ITGA2B P08514 6/20 0.47
ALDH1A1 P00352 1/20 0.45
LMNA P02545 1/20 0.45
HPGD P15428 1/20 0.45
AKR1C3 P42330 1/20 0.45
HTT P42858 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
USP2 O75604 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2C9 P11712 1/20 0.45
TSHR P16473 1/20 0.45
CYP2C19 P33261 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL745801 0.89 EPHX2 (0.52) EPHX2ITGB3ITGA2BAKR1C3
SCHEMBL747330 0.82 EPHX2 (0.51) EPHX2ITGB3ITGA2BALDH1A1HPGD
SCHEMBL743550 0.79 CYP3A4 (0.49) EPHX2ALDH1A1HPGDSMN1; SMN2USP2
SCHEMBL26552871 0.78 ALDH1A1 (0.47) EPHX2ALDH1A1
SCHEMBL743517 0.78 MAPK1 (0.54) EPHX2ITGB3ITGA2BALDH1A1HPGD
SCHEMBL3748988 0.78 LIPE (0.60) EPHX2
SCHEMBL3748578 0.78 LIPE (0.60) EPHX2
SCHEMBL5888 0.78 EPHX2 (0.49) EPHX2
SCHEMBL5019 0.78 SLC6A4 (0.49) EPHX2
SCHEMBL746449 0.77 EPHX2 (0.48) EPHX2ALDH1A1HPGDSMN1; SMN2USP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2430023-A1 AZACYCLIC SPIRODERIVATIVES AS HSL INHIBITORS F. Hoffmann-La Roche AG (CH) 2012-03-21 EP claimed
WO-2010130665-A1 AZACYCLIC SPIRODERIVATIVES AS HSL INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2010-11-18 WO claimed