SCHEMBL7478643

SCHEMBL7478643

CC(C)CC(NC(=O)COc1ccccc1C(C)(C)C)C(=O)NC(Cc1ccc(OC(=O)N2CCN(C(=O)c3ccccc3)CC2)cc1)C(=O)O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 3/20 0.44
ITGA4 P13612 3/20 0.44
ITGB7 P26010 2/20 0.44
CACNA1B Q00975 3/20 0.43
YAP1 P46937 3/20 0.42
GPR34 Q9UPC5 2/20 0.40
MAPK1 P28482 1/20 0.39
CASP1 P29466 4/20 0.39
CASP3 P42574 4/20 0.39
CASP7 P55210 4/20 0.39
CASP6 P55212 4/20 0.39
CASP8 Q14790 4/20 0.39
MEN1 O00255 1/20 0.38
ALDH1A1 P00352 1/20 0.38
LMNA P02545 1/20 0.38
KMT2A Q03164 1/20 0.38
MMP2 P08253 1/20 0.38
MMP7 P09237 1/20 0.38
MMP9 P14780 1/20 0.38
MMP12 P39900 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6473763 1.00 ITGB1 (0.44) ITGB1ITGA4ITGB7CACNA1BYAP1
SCHEMBL6474215 0.93 ITGB1 (0.46) ITGB1ITGA4ITGB7CACNA1BYAP1
SCHEMBL6474104 0.91 KMT2A (0.45) ITGB1ITGA4ITGB7CACNA1BYAP1
SCHEMBL6478996 0.91 CACNA1B (0.47) ITGB1ITGA4ITGB7CACNA1BYAP1
SCHEMBL6481231 0.90 ITGB1 (0.46) ITGB1ITGA4ITGB7CACNA1BYAP1
SCHEMBL6479143 0.90 ITGB1 (0.45) ITGB1ITGA4ITGB7CACNA1BYAP1
SCHEMBL6480951 0.89 MAPK1 (0.47) ITGB1ITGA4ITGB7CACNA1BYAP1
SCHEMBL6480791 0.87 YAP1 (0.46) ITGB1ITGA4ITGB7YAP1GPR34
SCHEMBL6474590 0.87 ITGB1 (0.49) ITGB1ITGA4ITGB7CACNA1BYAP1
SCHEMBL6481324 0.86 MAPK1 (0.44) ITGB1ITGA4ITGB7CACNA1BYAP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140837-A1 COMPOUNDS USEFUL IN THE TREATMENT OF INFLAMMATORY DISEASES GLAXO GROUP LIMITED (GB) 2001-10-10 EP disclosed
WO-2000037444-A1 COMPOUNDS USEFUL IN THE TREATMENT OF INFLAMMATORY DISEASES GLAXO GROUP LIMITED (GB) 2000-06-29 WO disclosed