SCHEMBL7479714

SCHEMBL7479714

O=C1c2ccccc2C(=O)N1Nc1ccccn1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.53
KDM4E B2RXH2 1/20 0.50
MEN1 O00255 3/20 0.48
KMT2A Q03164 3/20 0.48
ALDH1A1 P00352 3/20 0.48
NPSR1 Q6W5P4 1/20 0.48
PKM P14618 2/20 0.46
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
HSD17B10 Q99714 1/20 0.44
LMNA P02545 1/20 0.42
MAPK10 P53779 1/20 0.42
GFER P55789 1/20 0.42
GAA P10253 1/20 0.42
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
MAPK1 P28482 1/20 0.41
CHRNB2 P17787 1/20 0.41
CHRNB4 P30926 1/20 0.41
CHRNA3 P32297 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11196972 0.82 KDM4E (0.48) CYP1A2KDM4EMEN1KMT2AALDH1A1
SCHEMBL20515677 0.81 CYP1A2 (0.57) CYP1A2KDM4EMEN1KMT2AALDH1A1
SCHEMBL7485009 0.72 CYP1A2 (0.71) CYP1A2KDM4EALDH1A1NPC1RAB9A
SCHEMBL8812148 0.70 HPGD (0.41) KDM4EMEN1KMT2AALDH1A1NPSR1
SCHEMBL3259551 0.70 CYP1A2 (1.00) CYP1A2KDM4EMEN1KMT2AALDH1A1
SCHEMBL25215843 0.69 LMNA (0.60) CYP1A2KDM4EMEN1KMT2AALDH1A1
SCHEMBL7479419 0.68 ALDH1A1 (0.73) KDM4EMEN1KMT2AALDH1A1NPSR1
Hydrochloric Acid SCHEMBL5138493 0.68 CYP1A2 (0.96) CYP1A2KDM4EMEN1KMT2AALDH1A1
SCHEMBL30817653 0.68 ALDH1A1 (0.73) KDM4EMEN1KMT2AALDH1A1NPSR1
SCHEMBL6859755 0.68 MEN1 (0.48) CYP1A2KDM4EMEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0950056-B1 N-(PYRIDINYLAMINO)ISOINDOLINES AND RELATED COMPOUNDS AVENTIS PHARMA INC (US) 2002-09-18 EP disclosed
CN-1242012-A N- (pyridylamino) isoindolines and related compounds HOECHST MARION ROUSSEL INC (US) 2000-01-19 CN disclosed
US-6004977-A ANTIDEPRESSANTS, COGNITION ACTIVATORS, AND ALZHEIMER'S DISEASE TREATMENT HOECHST MARION ROUSSEL, INC. (US) 1999-12-21 US disclosed
EP-0950056-A2 N-(PYRIDINYLAMINO)ISOINDOLINES AND RELATED COMPOUNDS HOECHST MARION ROUSSEL, INC. (US) 1999-10-20 EP disclosed
WO-1998029407-A2 N-(PYRIDINYLAMINO)ISOINDOLINES FOR TREATING ALZHEIMER'S AND DEPRESSION HOECHST MARION ROUSSEL, INC. (US) 1998-07-09 WO disclosed