SCHEMBL7479968

SCHEMBL7479968

CC1(C)CC(=O)c2c(-c3ccncc3)n[nH]c2C1

nearest known ligand 0.73

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ALPL P05186 7/20 0.73
HSD17B10 Q99714 2/20 0.62
ALDH1A1 P00352 2/20 0.62
HPGD P15428 2/20 0.62
KDM4E B2RXH2 1/20 0.62
CYP3A4 P08684 1/20 0.50
CYP2C9 P11712 1/20 0.50
CYP2C19 P33261 1/20 0.50
BUB1 O43683 11/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7480743 0.82 ALPL (0.72) ALPLHSD17B10ALDH1A1HPGDKDM4E
SCHEMBL17977834 0.78 ALPL (0.70) ALPLHSD17B10ALDH1A1HPGDKDM4E
SCHEMBL7491199 0.76 ALPL (0.74) ALPLHSD17B10ALDH1A1HPGDKDM4E
SCHEMBL7490603 0.74 ALPL (0.64) ALPLHSD17B10ALDH1A1HPGDKDM4E
SCHEMBL7490668 0.74 ALPL (0.65) ALPLHSD17B10ALDH1A1HPGDKDM4E
SCHEMBL7482110 0.74 ALPL (0.58) ALPLHSD17B10ALDH1A1HPGDKDM4E
SCHEMBL7484888 0.73 ROCK2 (0.42) ALPLHSD17B10ALDH1A1HPGDKDM4E
SCHEMBL7684925 0.73 BUB1 (0.65) BUB1
SCHEMBL17372220 0.72 BUB1 (0.66) BUB1
SCHEMBL460286 0.72 HSD17B10 (0.63) ALPLHSD17B10ALDH1A1HPGDKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1177185-A1 4, 5, 6, 7-TETRAHYDROINDAZOLE DERIVATIVES AS ANTITUMOR AGENTS PHARMACIA & UPJOHN S.p.A. (IT) 2002-02-06 EP disclosed
WO-2000069846-A1 4,5,6,7-TETRAHYDROINDAZOLE DERIVATIVES AS ANTITUMOR AGENTS PHARMACIA & UPJOHN S.P.A. (IT) 2000-11-23 WO disclosed