SCHEMBL7480353

SCHEMBL7480353

O=C(O)Oc1cccc2[nH]c(-c3cnn(-c4ccc(Cl)cc4)c3)nc12

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 6/20 0.44
NR2E3 Q9Y5X4 1/20 0.43
MAP4K4 O95819 1/20 0.42
MGAM O43451 1/20 0.40
GAA P10253 1/20 0.40
SI P14410 1/20 0.40
MGAM2 Q2M2H8 1/20 0.40
HPSE Q9Y251 2/20 0.39
EGLN1 Q9GZT9 1/20 0.39
DHODH Q02127 4/20 0.37
DGAT2 Q96PD7 1/20 0.37
NPC1 O15118 1/20 0.36
MAPT P10636 1/20 0.36
NFKB1 P19838 1/20 0.36
RAB9A P51151 1/20 0.36
NFKB2 Q00653 1/20 0.36
RELA Q04206 1/20 0.36
PTGDR2 Q9Y5Y4 1/20 0.36
TNKS O95271 1/20 0.36
TNKS2 Q9H2K2 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6591596 0.91 PARP1 (0.48) PARP1NR2E3MAP4K4MGAMGAA
SCHEMBL6585150 0.83 PARP1 (0.46) PARP1NR2E3HPSEDHODHDGAT2
SCHEMBL6810606 0.81 PARP1 (0.69) PARP1MAP4K4DHODHPARP2
SCHEMBL6586796 0.81 PKN1 (0.39) PARP1NR2E3MAP4K4HPSEDHODH
SCHEMBL7478464 0.79 PARP1 (0.41) PARP1MGAMGAASIMGAM2
SCHEMBL12834073 0.74 AURKA (0.51) MAP4K4HPSEMAPT
SCHEMBL6587289 0.73 PARP1 (0.49) PARP1MAP4K4MGAMGAASI
SCHEMBL6806394 0.73 PARP1 (0.67) PARP1MAP4K4DHODHPARP2
SCHEMBL6591702 0.71 PARP1 (0.44) PARP1MAP4K4MGAMGAASI
SCHEMBL6590978 0.71 PARP1 (0.42) PARP1MGAMGAASIMGAM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1177178-A1 HETEROCYCLICALLY SUBSTITUTED BENZIMIDAZOLES, THE PRODUCTION AND APPLICATION THEREOF BASF AKTIENGESELLSCHAFT (DE) 2002-02-06 EP disclosed
WO-2001082877-A2 USE OF PARP INHIBITORS IN COSMETIC PREPARATIONS BASF AKTIENGESELLSCHAFT (DE) 2001-11-08 WO disclosed
WO-2000068206-A1 HETEROCYCLICALLY SUBSTITUTED BENZIMIDAZOLES, THE PRODUCTION AND APPLICATION THEREOF BASF AKTIENGESELLSCHAFT (DE) 2000-11-16 WO disclosed