SCHEMBL7478464

SCHEMBL7478464

O=C(O)Oc1cccc2[nH]c(-c3ccnn3-c3ccc(Cl)cc3)nc12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 4/20 0.41
NR3C2 P08235 1/20 0.37
GAA P10253 2/20 0.37
MGAM O43451 1/20 0.37
SI P14410 1/20 0.37
MGAM2 Q2M2H8 1/20 0.37
DHODH Q02127 3/20 0.36
PTGER1 P34995 1/20 0.36
HPSE Q9Y251 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
ADORA2B P29275 1/20 0.35
FFAR4 Q5NUL3 1/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
LMNA P02545 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
BRAF P15056 1/20 0.35
CBFB Q13951 2/20 0.34
ALDH1A1 P00352 1/20 0.34
TP53 P04637 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6591702 0.92 PARP1 (0.44) PARP1NR3C2GAAMGAMSI
SCHEMBL6807081 0.82 PARP1 (0.64) PARP1DHODH
SCHEMBL7480353 0.79 PARP1 (0.44) PARP1GAAMGAMSIMGAM2
SCHEMBL6585205 0.73 PARP1 (0.42) PARP1GAAMGAMSIMGAM2
SCHEMBL7480214 0.72 HPSE (0.38) PARP1DHODHHPSESMN1; SMN2CBFB
SCHEMBL6587560 0.71 PARP1 (0.42) PARP1GAAMGAMSIMGAM2
SCHEMBL6591596 0.70 PARP1 (0.48) PARP1GAAMGAMSIMGAM2
SCHEMBL6807085 0.70 NR3C2 (0.43) PARP1NR3C2MEN1KMT2AADORA2B
SCHEMBL6587289 0.69 PARP1 (0.49) PARP1GAAMGAMSIMGAM2
SCHEMBL12662069 0.68 DHODH (0.41) PARP1NR3C2DHODHADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1177178-A1 HETEROCYCLICALLY SUBSTITUTED BENZIMIDAZOLES, THE PRODUCTION AND APPLICATION THEREOF BASF AKTIENGESELLSCHAFT (DE) 2002-02-06 EP disclosed
WO-2001082877-A2 USE OF PARP INHIBITORS IN COSMETIC PREPARATIONS BASF AKTIENGESELLSCHAFT (DE) 2001-11-08 WO disclosed
WO-2000068206-A1 HETEROCYCLICALLY SUBSTITUTED BENZIMIDAZOLES, THE PRODUCTION AND APPLICATION THEREOF BASF AKTIENGESELLSCHAFT (DE) 2000-11-16 WO disclosed