SCHEMBL7480819

SCHEMBL7480819

Cc1cc(-c2nc(CS(=O)(=O)c3ccccc3)n[nH]2)oc1C

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.42
NPC1 O15118 6/20 0.39
RAB9A P51151 6/20 0.39
TDP1 Q9NUW8 2/20 0.39
SMN1; SMN2 Q16637 5/20 0.37
TSHR P16473 1/20 0.35
LMNA P02545 1/20 0.34
MAPT P10636 2/20 0.34
POLB P06746 2/20 0.34
HTT P42858 1/20 0.34
CYP2D6 P10635 1/20 0.34
HPGD P15428 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7482899 0.78 HPGD (0.48) ALDH1A1NPC1RAB9ATDP1SMN1; SMN2
SCHEMBL7484505 0.76 NR1H2 (0.46) ALDH1A1NPC1RAB9ASMN1; SMN2TSHR
SCHEMBL7482166 0.71 DCUN1D1 (0.48) ALDH1A1NPC1RAB9ATDP1SMN1; SMN2
SCHEMBL7425395 0.71 SMN1; SMN2 (0.50) ALDH1A1NPC1RAB9ATDP1SMN1; SMN2
SCHEMBL7434319 0.70 GRK6 (0.47) ALDH1A1NPC1RAB9ASMN1; SMN2LMNA
SCHEMBL7486751 0.70 ALOX5AP (0.38) ALDH1A1MAPTPOLB
SCHEMBL7487218 0.69 SMN1; SMN2 (0.51) NPC1SMN1; SMN2LMNAMAPTHTT
SCHEMBL7482611 0.69 PSIP1 (0.41) ALDH1A1NPC1RAB9ATDP1SMN1; SMN2
SCHEMBL7480824 0.65 TDP1 (0.35) ALDH1A1NPC1RAB9ATDP1SMN1; SMN2
SCHEMBL2069838 0.64 NPC1 (0.52) ALDH1A1NPC1RAB9ATDP1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1379777-A Amino-triazolopyridine derivatives HOFFMANN LA ROCHE (CH) 2002-11-13 CN disclosed
EP-1214322-A2 AMINO-TRIAZOLOPYRIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2002-06-19 EP disclosed
US-6355653-B1 DRUG AND CARRIER FOR ANTIALLERGENS, BRAIN DISORDERS AND NEUROTRANSMITTERS HOFFMANN-LA ROCHE INC. 2002-03-12 US disclosed
WO-2001017999-A2 AMINO-TRIAZOLOPYRIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2001-03-15 WO disclosed