SCHEMBL7480824

SCHEMBL7480824

Cc1cc(-c2ncnn2CS(=O)(=O)c2ccccc2)oc1C

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 3/20 0.35
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
PSIP1 O75475 1/20 0.34
ALDH1A1 P00352 4/20 0.33
SMN1; SMN2 Q16637 3/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
HSD11B1 P28845 1/20 0.32
USP2 O75604 1/20 0.32
GAA P10253 1/20 0.32
FLT1 P17948 1/20 0.32
FLT4 P35916 1/20 0.32
KDR P35968 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.31
POLB P06746 2/20 0.31
APLNR P35414 1/20 0.31
MAPT P10636 1/20 0.31
LMNA P02545 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7484993 0.79 ALDH1A1 (0.42) TDP1NPC1RAB9AALDH1A1SMN1; SMN2
SCHEMBL7490899 0.77 HDAC1 (0.45) TDP1NPC1RAB9APSIP1ALDH1A1
SCHEMBL7481950 0.73 ALDH1A1 (0.38) NPC1RAB9APSIP1ALDH1A1SMN1; SMN2
SCHEMBL7487578 0.72 HDAC1 (0.48) TDP1NPC1RAB9APSIP1POLB
SCHEMBL7482230 0.71 HDAC1 (0.47) ALDH1A1SMN1; SMN2MEN1KMT2AUSP2
SCHEMBL7486763 0.71 NSD2 (0.39) HSD11B1
SCHEMBL7487226 0.70 PTGS2 (0.40) ALDH1A1SMN1; SMN2HSD11B1L3MBTL1
SCHEMBL7482618 0.70 PSIP1 (0.41) NPC1RAB9APSIP1ALDH1A1SMN1; SMN2
SCHEMBL7480819 0.65 ALDH1A1 (0.42) TDP1NPC1RAB9AALDH1A1SMN1; SMN2
SCHEMBL347966 0.60 MAOB (0.53) TDP1NPC1RAB9AALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1214322-A2 AMINO-TRIAZOLOPYRIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2002-06-19 EP disclosed
US-6355653-B1 DRUG AND CARRIER FOR ANTIALLERGENS, BRAIN DISORDERS AND NEUROTRANSMITTERS HOFFMANN-LA ROCHE INC. 2002-03-12 US disclosed
WO-2001017999-A2 AMINO-TRIAZOLOPYRIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2001-03-15 WO disclosed