SCHEMBL7480917

SCHEMBL7480917

CCCCCNc1cnc(-c2ccc(OC(F)(F)F)cc2OC)c(OC)n1

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CRHR1 P34998 9/20 0.51
SCN9A Q15858 1/20 0.40
RUNX1 Q01196 1/20 0.40
ADORA3 P0DMS8 2/20 0.36
PIM1 P11309 1/20 0.35
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
HPGD P15428 1/20 0.35
TSHR P16473 1/20 0.35
MAPK1 P28482 1/20 0.35
HSD17B10 Q99714 1/20 0.35
ABL1 P00519 1/20 0.34
MERTK Q12866 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6201263 0.84 CRHR1 (0.62) CRHR1SCN9A
SCHEMBL5417862 0.83 CRHR1 (0.49) CRHR1SCN9ARUNX1PIM1HPGD
SCHEMBL7473622 0.82 CRHR1 (0.58) CRHR1SCN9A
SCHEMBL7476681 0.82 CRHR1 (0.58) CRHR1SCN9AADORA3ALDH1A1
SCHEMBL5420406 0.82 CRHR1 (0.68) CRHR1SCN9ARUNX1
SCHEMBL6203614 0.82 CRHR1 (0.70) CRHR1SCN9A
SCHEMBL5409112 0.81 CRHR1 (0.50) CRHR1SCN9ARUNX1ABL1
SCHEMBL6201786 0.77 CRHR1 (0.60) CRHR1SCN9A
SCHEMBL5417192 0.76 CRHR1 (0.62) CRHR1SCN9ARUNX1
SCHEMBL4924779 0.76 CRHR1 (0.58) CRHR1SCN9AADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1255740-A2 SUBSTITUTED ARYLPYRAZINES NEUROGEN CORPORATION (US) 2002-11-13 EP disclosed
WO-2001060806-A2 SUBSTITUTED ARYLPYRAZINES NEUROGEN CORPORATION (US) 2001-08-23 WO disclosed