SCHEMBL7480938

SCHEMBL7480938

Oc1ccc2c(c1)CN(Nc1ccccn1)C2

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.43
RAB9A P51151 4/20 0.43
MEN1 O00255 4/20 0.43
KMT2A Q03164 4/20 0.43
NCOA1 Q15788 1/20 0.41
NCOA3 Q9Y6Q9 1/20 0.41
STAT3 P40763 1/20 0.40
STAT1 P42224 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
PKM P14618 1/20 0.37
POLB P06746 2/20 0.36
DRD1 P21728 1/20 0.36
DRD5 P21918 1/20 0.36
HSP90AA1 P07900 1/20 0.36
HSP90AB1 P08238 1/20 0.36
PDK2 Q15119 1/20 0.35
GAA P10253 3/20 0.35
ESR2 Q92731 1/20 0.35
KCNMA1 Q12791 1/20 0.35
MIF P14174 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7480356 0.99 NPC1 (0.42) NPC1RAB9AMEN1KMT2ANCOA1
SCHEMBL7474257 0.84 MEN1 (0.44) NPC1RAB9AMEN1KMT2ASMN1; SMN2
SCHEMBL27528778 0.77 GRIN2B (0.39) NPC1RAB9AMEN1KMT2APKM
SCHEMBL7481791 0.77 ALDH1A1 (0.41) NPC1RAB9AMEN1KMT2ASTAT3
SCHEMBL7480814 0.76 KMT2A (0.46) NPC1RAB9AMEN1KMT2ASMN1; SMN2
SCHEMBL7482791 0.76 MAPK1 (0.41) NPC1RAB9AMEN1KMT2ASMN1; SMN2
SCHEMBL7480818 0.75 ALDH1A1 (0.47) NPC1RAB9ASMN1; SMN2PKMALDH1A1
SCHEMBL7482069 0.74 NPC1 (0.36) NPC1RAB9AMEN1KMT2ASMN1; SMN2
SCHEMBL7481558 0.74 CYP19A1 (0.41) DRD1DRD5PDK2ESR2ESR1
SCHEMBL7480185 0.74 GRIN2D (0.51) KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0950056-B1 N-(PYRIDINYLAMINO)ISOINDOLINES AND RELATED COMPOUNDS AVENTIS PHARMA INC (US) 2002-09-18 EP claimed
CN-1242012-A N- (pyridylamino) isoindolines and related compounds HOECHST MARION ROUSSEL INC (US) 2000-01-19 CN claimed
EP-0950056-A2 N-(PYRIDINYLAMINO)ISOINDOLINES AND RELATED COMPOUNDS HOECHST MARION ROUSSEL, INC. (US) 1999-10-20 EP claimed
WO-1998029407-A2 N-(PYRIDINYLAMINO)ISOINDOLINES FOR TREATING ALZHEIMER'S AND DEPRESSION HOECHST MARION ROUSSEL, INC. (US) 1998-07-09 WO claimed
EP-0950056-B1 N-(PYRIDINYLAMINO)ISOINDOLINES AND RELATED COMPOUNDS AVENTIS PHARMA INC (US) 2002-09-18 EP disclosed
CN-1242012-A N- (pyridylamino) isoindolines and related compounds HOECHST MARION ROUSSEL INC (US) 2000-01-19 CN disclosed
US-6004977-A ANTIDEPRESSANTS, COGNITION ACTIVATORS, AND ALZHEIMER'S DISEASE TREATMENT HOECHST MARION ROUSSEL, INC. (US) 1999-12-21 US disclosed
EP-0950056-A2 N-(PYRIDINYLAMINO)ISOINDOLINES AND RELATED COMPOUNDS HOECHST MARION ROUSSEL, INC. (US) 1999-10-20 EP disclosed
WO-1998029407-A2 N-(PYRIDINYLAMINO)ISOINDOLINES FOR TREATING ALZHEIMER'S AND DEPRESSION HOECHST MARION ROUSSEL, INC. (US) 1998-07-09 WO disclosed