SCHEMBL7482154

SCHEMBL7482154

Nc1sc2c(c1C(=O)O)CCOC2CO

nearest known ligand 0.37

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 3/20 0.37
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
MAPT P10636 1/20 0.37
RAD52 P43351 1/20 0.37
PTPN2 P17706 1/20 0.35
PTPN1 P18031 1/20 0.35
PTPRB P23467 1/20 0.35
DRD1 P21728 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5838350 0.81 ADORA1 (0.38) ADORA1KDM4EALDH1A1MAPT
SCHEMBL5837036 0.78 PTPN1 (0.55) PTPN2PTPN1PTPRB
SCHEMBL7490616 0.77 ALDH1A1 (0.34) ADORA1KDM4EALDH1A1MAPTRAD52
SCHEMBL7861190 0.76 CYP1A2 (0.42) ADORA1KDM4EALDH1A1PTPN2PTPN1
SCHEMBL7536578 0.74 PTPN1 (0.38) PTPN2PTPN1PTPRB
SCHEMBL7482552 0.72 KDM4E (0.34) ADORA1KDM4EALDH1A1MAPTRAD52
SCHEMBL5838672 0.70 ADORA1 (0.38) ADORA1KDM4EALDH1A1MAPTDRD1
SCHEMBL7486653 0.70 ADORA1 (0.43) ADORA1ALDH1A1MAPT
SCHEMBL27558405 0.67 ALDH1A1 (0.43) ADORA1KDM4EALDH1A1MAPTRAD52
SCHEMBL6317021 0.67 ADORA1 (0.35) ADORA1KDM4EALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1214060-A2 METHOD OF INHIBITING PROTEIN TYROSINE PHOSPHATASE 1B AND/OR T-CELL PROTEIN TYROSINE PHOSPHATASE AND/OR OTHER PTPASES WITH AN ASP RESIDUE AT POSITION 48 NOVO NORDISK A/S (DK) 2002-06-19 EP disclosed
WO-2001017516-A2 METHOD OF INHIBITING PROTEIN TYROSINE PHOSPHATASE 1B AND/OR T-CELL PROTEIN TYROSINE PHOSPHATASE AND/OR OTHER PTPASES WITH AN ASP RESIDUE AT POSITION 48 NOVO NORDISK A/S (DK) 2001-03-15 WO disclosed