SCHEMBL7485013

SCHEMBL7485013

O=C(O)Oc1cccc2[nH]c(-c3ccc(N4CCNCC4)nc3)nc12

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
AURKA O14965 2/20 0.52
AURKB Q96GD4 2/20 0.52
KDR P35968 1/20 0.52
DGAT1 O75907 10/20 0.51
KCNH2 Q12809 9/20 0.51
ADORA2A P29274 6/20 0.51
PRMT5 O14744 2/20 0.42
PARP1 P09874 3/20 0.41
HPSE Q9Y251 1/20 0.41
CDK1 P06493 1/20 0.41
CDK2 P24941 1/20 0.41
MKNK1 Q9BUB5 1/20 0.41
MKNK2 Q9HBH9 1/20 0.41
CACNA1C Q13936 1/20 0.40
ASIC3 Q9UHC3 1/20 0.40
DHODH Q02127 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7759237 0.92 AURKA (0.54) AURKAAURKBKDRDGAT1KCNH2
SCHEMBL6588365 0.91 AURKA (0.54) AURKAAURKBKDRDGAT1KCNH2
SCHEMBL7480315 0.91 AURKA (0.53) AURKAAURKBKDRDGAT1KCNH2
SCHEMBL6591285 0.88 AURKA (0.51) AURKAAURKBKDRDGAT1KCNH2
SCHEMBL6587264 0.83 AURKA (0.55) AURKAAURKBKDRDGAT1KCNH2
SCHEMBL6587278 0.82 AURKA (0.54) AURKAAURKBKDRDGAT1KCNH2
SCHEMBL6587512 0.82 AURKA (0.54) AURKAAURKBKDRDGAT1KCNH2
SCHEMBL6805718 0.82 AURKA (0.72) AURKAAURKBKDRPARP1DHODH
SCHEMBL6586056 0.82 AURKA (0.59) AURKAAURKBKDRDGAT1KCNH2
SCHEMBL6590217 0.80 AURKA (0.59) AURKAAURKBKDRDGAT1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1177178-A1 HETEROCYCLICALLY SUBSTITUTED BENZIMIDAZOLES, THE PRODUCTION AND APPLICATION THEREOF BASF AKTIENGESELLSCHAFT (DE) 2002-02-06 EP disclosed
WO-2001082877-A2 USE OF PARP INHIBITORS IN COSMETIC PREPARATIONS BASF AKTIENGESELLSCHAFT (DE) 2001-11-08 WO disclosed
WO-2000068206-A1 HETEROCYCLICALLY SUBSTITUTED BENZIMIDAZOLES, THE PRODUCTION AND APPLICATION THEREOF BASF AKTIENGESELLSCHAFT (DE) 2000-11-16 WO disclosed