SCHEMBL7485182

SCHEMBL7485182

COc1ccc(-c2cc(N)n3nc(-c4ccccn4)nc3c2)nc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 1/20 0.49
F2 P00734 1/20 0.47
F12 P00748 1/20 0.47
SMN1; SMN2 Q16637 7/20 0.45
NPC1 O15118 6/20 0.45
RAB9A P51151 6/20 0.45
ALDH1A1 P00352 4/20 0.45
PKM P14618 3/20 0.45
ATM Q13315 3/20 0.45
KDM4E B2RXH2 1/20 0.45
HPGD P15428 1/20 0.45
CDK5 Q00535 1/20 0.45
CDK5R1 Q15078 1/20 0.45
L3MBTL1 Q9Y468 4/20 0.42
HSP90AA1 P07900 1/20 0.42
LMNA P02545 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
GRM5 P41594 1/20 0.40
FFAR1 O14842 1/20 0.39
PIK3CA P42336 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7431382 0.89 NPC1 (0.52) ADORA2AF2F12SMN1; SMN2NPC1
SCHEMBL7428533 0.87 ADORA2A (0.60) ADORA2AF2F12SMN1; SMN2NPC1
SCHEMBL7483006 0.85 NPC1 (0.53) ADORA2AF2F12SMN1; SMN2NPC1
SCHEMBL7426124 0.84 ADORA2A (0.51) ADORA2AF2F12SMN1; SMN2NPC1
SCHEMBL7703002 0.84 ADORA2A (0.47) ADORA2AF2F12SMN1; SMN2NPC1
SCHEMBL7434316 0.84 ADORA2A (0.48) ADORA2AF2F12SMN1; SMN2NPC1
SCHEMBL7709217 0.81 GRM5 (0.50) ADORA2AF2F12SMN1; SMN2NPC1
SCHEMBL7709212 0.80 ADORA2A (0.49) ADORA2ANPC1ALDH1A1ATMKDM4E
SCHEMBL7542178 0.80 ADORA2A (0.52) ADORA2ASMN1; SMN2NPC1RAB9AALDH1A1
SCHEMBL7708845 0.78 ADORA2A (0.54) ADORA2AF2F12SMN1; SMN2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1214322-A2 AMINO-TRIAZOLOPYRIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2002-06-19 EP disclosed
WO-2001017999-A2 AMINO-TRIAZOLOPYRIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2001-03-15 WO disclosed