SCHEMBL7485306

SCHEMBL7485306

COc1cc2nccc(Oc3ccc(C(=O)c4cccc(F)c4)cc3)c2cc1OC

nearest known ligand 0.69

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
FGFR2 P21802 2/20 0.69
KDR P35968 12/20 0.67
PDGFRA P16234 12/20 0.67
SRC P12931 1/20 0.59
TGFBR1 P36897 1/20 0.59
KIT P10721 1/20 0.57
AXL P30530 1/20 0.57
MET P08581 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7487173 0.90 FGFR2 (0.76) FGFR2KDRPDGFRASRCTGFBR1
SCHEMBL7487378 0.89 FGFR2 (0.77) FGFR2KDRPDGFRASRCTGFBR1
SCHEMBL3905120 0.88 FGFR2 (0.70) FGFR2KDRPDGFRASRCTGFBR1
SCHEMBL7482200 0.87 FGFR2 (0.69) FGFR2KDRPDGFRASRCTGFBR1
SCHEMBL7485632 0.87 FGFR2 (0.71) FGFR2KDRPDGFRASRCTGFBR1
SCHEMBL7485757 0.85 FGFR2 (0.71) FGFR2KDRPDGFRASRCTGFBR1
SCHEMBL3901338 0.84 SRC (0.70) FGFR2KDRPDGFRASRCTGFBR1
SCHEMBL7481918 0.84 FGFR2 (0.77) FGFR2KDRPDGFRASRCTGFBR1
SCHEMBL7482945 0.84 FGFR2 (0.72) FGFR2KDRPDGFRASRCTGFBR1
SCHEMBL7482801 0.83 FGFR2 (0.76) FGFR2KDRPDGFRASRCTGFBR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0860433-B1 QUINOLINE DERIVATIVES AND QUINAZOLINE DERIVATIVES INHIBITING AUTOPHOSPHORYLATION OF GROWTH FACTOR RECEPTOR ORIGINATING IN PLATELET AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME KIRIN BREWERY (JP) 2002-07-03 EP disclosed
EP-0860433-A1 QUINOLINE DERIVATIVES AND QUINAZOLINE DERIVATIVES INHIBITING AUTOPHOSPHORYLATION OF GROWTH FACTOR RECEPTOR ORIGINATING IN PLATELET AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME KIRIN BEER KABUSHIKI KAISHA (JP) 1998-08-26 EP disclosed