SCHEMBL7485757

SCHEMBL7485757

COc1cc2nccc(Oc3ccc(C(=O)c4ccc5ccccc5c4)cc3)c2cc1OC

nearest known ligand 0.71

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
FGFR2 P21802 2/20 0.71
PDGFRA P16234 8/20 0.62
KDR P35968 8/20 0.62
SRC P12931 3/20 0.61
TGFBR1 P36897 3/20 0.61
MET P08581 3/20 0.59
AURKA O14965 2/20 0.59
LCK P06239 2/20 0.59
TEK Q02763 2/20 0.59
AURKB Q96GD4 2/20 0.59
KIT P10721 2/20 0.59
AXL P30530 1/20 0.59
ABL1 P00519 1/20 0.59
LYN P07948 1/20 0.59
PDGFRB P09619 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7487378 0.91 FGFR2 (0.77) FGFR2PDGFRAKDRSRCTGFBR1
SCHEMBL7482945 0.88 FGFR2 (0.72) FGFR2PDGFRAKDRSRCTGFBR1
SCHEMBL7481918 0.86 FGFR2 (0.77) FGFR2PDGFRAKDRSRCTGFBR1
SCHEMBL3905120 0.86 FGFR2 (0.70) FGFR2PDGFRAKDRSRCTGFBR1
SCHEMBL7482620 0.85 FGFR2 (0.76) FGFR2PDGFRAKDRSRCTGFBR1
SCHEMBL7482801 0.85 FGFR2 (0.76) FGFR2PDGFRAKDRSRCTGFBR1
SCHEMBL8069147 0.85 FGFR2 (0.76) FGFR2PDGFRAKDRSRCTGFBR1
SCHEMBL7487173 0.85 FGFR2 (0.76) FGFR2PDGFRAKDRSRCTGFBR1
SCHEMBL7482200 0.85 FGFR2 (0.69) FGFR2PDGFRAKDRSRCTGFBR1
SCHEMBL7485306 0.85 FGFR2 (0.69) FGFR2PDGFRAKDRSRCTGFBR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0860433-B1 QUINOLINE DERIVATIVES AND QUINAZOLINE DERIVATIVES INHIBITING AUTOPHOSPHORYLATION OF GROWTH FACTOR RECEPTOR ORIGINATING IN PLATELET AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME KIRIN BREWERY (JP) 2002-07-03 EP disclosed
US-6143764-A ETHER DERIVATIVES OF QUINOLINE, ANTITUMOR AGENTS KIRIN BEER KABUSHIKI KAISHA (JP) 2000-11-07 US disclosed
EP-0860433-A1 QUINOLINE DERIVATIVES AND QUINAZOLINE DERIVATIVES INHIBITING AUTOPHOSPHORYLATION OF GROWTH FACTOR RECEPTOR ORIGINATING IN PLATELET AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME KIRIN BEER KABUSHIKI KAISHA (JP) 1998-08-26 EP disclosed