SCHEMBL7487173

SCHEMBL7487173

COc1cc2nccc(Oc3ccc(C(=O)c4ccc(F)cc4)cc3)c2cc1OC

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FGFR2 P21802 2/20 0.76
PDGFRA P16234 10/20 0.74
KDR P35968 9/20 0.74
MET P08581 4/20 0.69
KIT P10721 2/20 0.66
AXL P30530 2/20 0.66
SRC P12931 2/20 0.66
AURKA O14965 1/20 0.66
RIPK2 O43353 1/20 0.66
ABCB11 O95342 1/20 0.66
ABL1 P00519 1/20 0.66
EGFR P00533 1/20 0.66
ERBB2 P04626 1/20 0.66
NTRK1 P04629 1/20 0.66
LCK P06239 1/20 0.66
PGR P06401 1/20 0.66
LYN P07948 1/20 0.66
RET P07949 1/20 0.66
CHRM2 P08172 1/20 0.66
HCK P08631 1/20 0.66

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7485306 0.90 FGFR2 (0.69) FGFR2PDGFRAKDRMETKIT
SCHEMBL7481918 0.89 FGFR2 (0.77) FGFR2PDGFRAKDRMETSRC
SCHEMBL7487378 0.89 FGFR2 (0.77) FGFR2PDGFRAKDRMETKIT
SCHEMBL7482620 0.88 FGFR2 (0.76) FGFR2PDGFRAKDRMETKIT
SCHEMBL8069147 0.88 FGFR2 (0.76) FGFR2PDGFRAKDRAXLSRC
SCHEMBL7482801 0.88 FGFR2 (0.76) FGFR2PDGFRAKDRMETKIT
SCHEMBL7486951 0.87 FGFR2 (0.74) FGFR2PDGFRAKDRMETKIT
SCHEMBL7485745 0.87 FGFR2 (0.82) FGFR2PDGFRAKDRMETSRC
SCHEMBL7482945 0.86 FGFR2 (0.72) FGFR2PDGFRAKDRMETKIT
SCHEMBL29574069 0.86 FGFR2 (1.00) FGFR2PDGFRAKDRMETKIT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0860433-B1 QUINOLINE DERIVATIVES AND QUINAZOLINE DERIVATIVES INHIBITING AUTOPHOSPHORYLATION OF GROWTH FACTOR RECEPTOR ORIGINATING IN PLATELET AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME KIRIN BREWERY (JP) 2002-07-03 EP disclosed
US-6143764-A ETHER DERIVATIVES OF QUINOLINE, ANTITUMOR AGENTS KIRIN BEER KABUSHIKI KAISHA (JP) 2000-11-07 US disclosed
EP-0860433-A1 QUINOLINE DERIVATIVES AND QUINAZOLINE DERIVATIVES INHIBITING AUTOPHOSPHORYLATION OF GROWTH FACTOR RECEPTOR ORIGINATING IN PLATELET AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME KIRIN BEER KABUSHIKI KAISHA (JP) 1998-08-26 EP disclosed