SCHEMBL7485337

SCHEMBL7485337

Cc1cc(-c2nc3cc(-c4ccncc4)cc(N)n3n2)oc1C

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 12/20 0.40
ALDH1A1 P00352 3/20 0.36
KDM4E B2RXH2 2/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
LMNA P02545 1/20 0.36
TP53 P04637 1/20 0.36
MAPT P10636 1/20 0.36
CYP2C19 P33261 1/20 0.36
NPC1 O15118 2/20 0.35
HPGD P15428 2/20 0.35
RAB9A P51151 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
NFKB1 P19838 1/20 0.35
HTT P42858 1/20 0.35
NFKB2 Q00653 1/20 0.35
RELA Q04206 1/20 0.35
GAA P10253 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7705907 0.84 ADORA2A (0.56) ADORA2AALDH1A1KDM4EMEN1KMT2A
SCHEMBL7711617 0.80 ADORA2A (0.44) ADORA2AALDH1A1KDM4ELMNAMAPT
SCHEMBL7430360 0.78 ADORA2A (0.56) ADORA2A
SCHEMBL7535250 0.77 ADORA2A (0.42) ADORA2A
SCHEMBL7427474 0.76 SMN1; SMN2 (0.47) ADORA2AALDH1A1KDM4EMEN1KMT2A
SCHEMBL7491116 0.76 ALDH1A1 (0.39) ADORA2AALDH1A1KDM4EMEN1KMT2A
SCHEMBL7711750 0.73 ADORA2A (0.57) ADORA2AALDH1A1KDM4EMEN1KMT2A
SCHEMBL7711685 0.73 ADORA2A (0.57) ADORA2AALDH1A1KDM4EMEN1KMT2A
SCHEMBL7709236 0.72 ALDH1A1 (0.48) ADORA2AALDH1A1KDM4EMEN1KMT2A
SCHEMBL7432234 0.72 ADORA2A (0.56) ADORA2AALDH1A1KDM4EMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1214322-A2 AMINO-TRIAZOLOPYRIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2002-06-19 EP disclosed
US-6355653-B1 DRUG AND CARRIER FOR ANTIALLERGENS, BRAIN DISORDERS AND NEUROTRANSMITTERS HOFFMANN-LA ROCHE INC. 2002-03-12 US disclosed
WO-2001017999-A2 AMINO-TRIAZOLOPYRIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2001-03-15 WO disclosed