SCHEMBL7427474

SCHEMBL7427474

Nc1cc(-c2ccncc2)cc2nc(-c3ccccc3)nn12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 6/20 0.47
NPC1 O15118 4/20 0.47
RAB9A P51151 4/20 0.47
ALDH1A1 P00352 3/20 0.47
HPGD P15428 2/20 0.47
NFKB1 P19838 2/20 0.47
NFKB2 Q00653 2/20 0.47
RELA Q04206 2/20 0.47
HTT P42858 1/20 0.47
KDM4E B2RXH2 2/20 0.44
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
MAPT P10636 2/20 0.44
GAA P10253 1/20 0.44
NOTUM Q6P988 1/20 0.43
ADORA3 P0DMS8 3/20 0.41
ADORA2A P29274 2/20 0.40
HSD17B10 Q99714 1/20 0.40
PDE10A Q9Y233 2/20 0.39
ADORA1 P30542 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7423524 0.93 ALDH1A1 (0.53) SMN1; SMN2NPC1RAB9AALDH1A1HPGD
SCHEMBL7426447 0.86 ADORA3 (0.46) SMN1; SMN2NPC1RAB9AALDH1A1HPGD
SCHEMBL7431418 0.84 ADORA2A (0.56) SMN1; SMN2NPC1RAB9AALDH1A1HPGD
SCHEMBL7709122 0.83 MAOA (0.47) SMN1; SMN2NPC1RAB9AALDH1A1HPGD
SCHEMBL7427040 0.83 NPC1 (0.42) SMN1; SMN2NPC1RAB9AALDH1A1HPGD
SCHEMBL7432234 0.81 ADORA2A (0.56) SMN1; SMN2NPC1RAB9AALDH1A1HPGD
SCHEMBL7708784 0.81 SMN1; SMN2 (0.54) SMN1; SMN2NPC1RAB9AALDH1A1HPGD
SCHEMBL7542178 0.81 ADORA2A (0.52) SMN1; SMN2NPC1RAB9AALDH1A1HPGD
SCHEMBL7703064 0.81 ALDH1A1 (0.45) SMN1; SMN2NPC1RAB9AALDH1A1HPGD
SCHEMBL7430360 0.80 ADORA2A (0.56) ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1214322-A2 AMINO-TRIAZOLOPYRIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2002-06-19 EP disclosed
US-6355653-B1 DRUG AND CARRIER FOR ANTIALLERGENS, BRAIN DISORDERS AND NEUROTRANSMITTERS HOFFMANN-LA ROCHE INC. 2002-03-12 US disclosed
WO-2001017999-A2 AMINO-TRIAZOLOPYRIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2001-03-15 WO disclosed