SCHEMBL7485387

SCHEMBL7485387

CC(C)(C)OC(=O)N1Cc2ccccc2C[C@H]1C(=O)NC[C@H](O)Cc1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 9/20 0.56
PTPN1 P18031 2/20 0.54
CXCR3 P49682 4/20 0.47
NPSR1 Q6W5P4 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7485383 1.00 HDAC8 (0.56) HDAC8PTPN1CXCR3NPSR1
SCHEMBL6238826 0.85 HDAC8 (0.70) HDAC8PTPN1CXCR3NPSR1
SCHEMBL22962123 0.83 MAPK1 (0.53) HDAC8PTPN1
SCHEMBL22962122 0.81 FNTA (0.51) HDAC8PTPN1NPSR1
SCHEMBL9033407 0.80 HDAC8 (0.53) HDAC8PTPN1
SCHEMBL9033397 0.80 HDAC8 (0.53) HDAC8PTPN1
SCHEMBL7479393 0.80 OPRM1 (0.55) HDAC8
SCHEMBL7479387 0.80 OPRM1 (0.55) HDAC8
SCHEMBL11986410 0.79 HDAC8 (0.53) HDAC8PTPN1CXCR3
SCHEMBL9033831 0.78 HDAC8 (0.64) HDAC8PTPN1CXCR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0914332-B1 ISOQUINOLINES USEFUL AS ANALGESICS ASTRAZENECA AB (SE) 2002-05-08 EP disclosed
US-6034097-A Isoquinolines useful as analgesics ASTRA AB (SE) 2000-03-07 US disclosed