SCHEMBL7486159

SCHEMBL7486159

O=C(c1ccc(O)cc1)C1CCCCC1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SRD5A2 P31213 1/20 0.65
MGLL Q99685 3/20 0.53
CNR1 P21554 1/20 0.47
CNR2 P34972 1/20 0.47
MIF P14174 2/20 0.46
DEGS1 O15121 1/20 0.46
RAB9A P51151 2/20 0.46
HRH3 Q9Y5N1 1/20 0.45
LMNA P02545 2/20 0.44
HTT P42858 2/20 0.44
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
ESR1 P03372 1/20 0.44
ESR2 Q92731 1/20 0.44
MAPT P10636 1/20 0.44
PKM P14618 1/20 0.44
HPGD P15428 1/20 0.44
NPC1 O15118 1/20 0.44
CYP2D6 P10635 1/20 0.44
ALDH1A1 P00352 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9136087 1.00 SRD5A2 (0.65) SRD5A2MGLLCNR1CNR2MIF
SCHEMBL1334288 0.98 SRD5A2 (0.61) SRD5A2MGLLCNR1CNR2MIF
SCHEMBL1335827 0.94 SRD5A2 (0.56) SRD5A2MGLLMIFRAB9ALMNA
SCHEMBL1334195 0.89 MGLL (0.57) SRD5A2MGLLRAB9ALMNAHTT
SCHEMBL5370523 0.89 MGLL (0.57) SRD5A2MGLLRAB9ALMNAHTT
SCHEMBL5370517 0.89 MGLL (0.57) SRD5A2MGLLRAB9ALMNAHTT
Water SCHEMBL6848223 0.85 MGLL (0.54) SRD5A2MGLLRAB9ALMNAHTT
SCHEMBL5460665 0.83 SRD5A2 (0.89) SRD5A2RAB9AHRH3LMNAHTT
SCHEMBL3161623 0.82 SRD5A2 (0.62) SRD5A2MGLLCNR1CNR2RAB9A
SCHEMBL507614 0.82 KMT2A (0.66) SRD5A2MGLLRAB9ALMNAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6441177-B1 Tertiary amines HOFFMANN-LA ROCHE INC. 2002-08-27 US disclosed
EP-0860433-B1 QUINOLINE DERIVATIVES AND QUINAZOLINE DERIVATIVES INHIBITING AUTOPHOSPHORYLATION OF GROWTH FACTOR RECEPTOR ORIGINATING IN PLATELET AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME KIRIN BREWERY (JP) 2002-07-03 EP disclosed
EP-0778264-B1 Tertiary amines having antimycotic and cholesterol lowering activity HOFFMANN LA ROCHE (CH) 2001-07-11 EP disclosed
US-6248765-B1 ANTIINFLAMMATORY AGENTS; HYPOTENSIVE AGENTS INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICAL (FR) 2001-06-19 US disclosed
US-6143764-A ETHER DERIVATIVES OF QUINOLINE, ANTITUMOR AGENTS KIRIN BEER KABUSHIKI KAISHA (JP) 2000-11-07 US disclosed
US-6034275-A FUGICIDES; ATICHOLESTEROL AGENTS HOFFMANN-LA ROCHE INC. (US) 2000-03-07 US disclosed
EP-0860433-A1 QUINOLINE DERIVATIVES AND QUINAZOLINE DERIVATIVES INHIBITING AUTOPHOSPHORYLATION OF GROWTH FACTOR RECEPTOR ORIGINATING IN PLATELET AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME KIRIN BEER KABUSHIKI KAISHA (JP) 1998-08-26 EP disclosed
EP-0778264-A1 Tertiary amines having antimycotic and cholesterol lowering activity F. HOFFMANN-LA ROCHE AG (CH) 1997-06-11 EP disclosed
US-5399698-A Lipoxygenase inhibitor intermediates BAYER AKTIENGESELLSCHAFT (DE) 1995-03-21 US disclosed
US-5231103-A Lipoxygenase inhibitors as antiinflammatory agents, antiasthma and cardiovascular disorders BAYER AKTIENGESELLSCHAFT (DE) 1993-07-27 US disclosed
EP-0525571-A1 Quinolin-2-yl-methoxybenzylhydroxyureas as lipoxygenase inhibitors BAYER AG (DE) 1993-02-03 EP disclosed
US-3979456-A Phenoxyalkylamines, process for their preparation and applications thereof LABORATOIRES LAROCHE NAVARRON (FR) 1976-09-07 US disclosed