SCHEMBL7486375

SCHEMBL7486375

COCC(COC)NC(c1ccccc1)(c1ccccc1)c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNN4 O15554 3/20 0.44
MAPT P10636 1/20 0.40
KIF11 P52732 2/20 0.37
NR1H2 P55055 1/20 0.35
NR1H3 Q13133 1/20 0.35
MAPK1 P28482 1/20 0.34
KDM4E B2RXH2 3/20 0.33
LMNA P02545 2/20 0.33
ALDH1A1 P00352 2/20 0.33
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA3 P07451 1/20 0.33
CA4 P22748 1/20 0.33
CA6 P23280 1/20 0.33
CA5A P35218 1/20 0.33
CA7 P43166 1/20 0.33
CACNA1C Q13936 1/20 0.33
SCN9A Q15858 1/20 0.33
CA9 Q16790 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14613732 0.83 KCNN4 (0.42) KCNN4MAPTKIF11KDM4EALDH1A1
SCHEMBL2552945 0.81 KCNN4 (0.35) KCNN4MAPTKIF11KDM4ECACNA1C
SCHEMBL8214268 0.80 CHRM3 (0.40) KCNN4MAPTKIF11KDM4ELMNA
SCHEMBL225196 0.78 CA12 (0.44) KCNN4MAPTKIF11KDM4ELMNA
SCHEMBL7418701 0.74 KCNN4 (0.35) KCNN4MAPTKIF11KDM4ELMNA
SCHEMBL7479981 0.74 KCNN4 (0.43) KCNN4MAPTKIF11MAPK1KDM4E
SCHEMBL8945099 0.73 KCNN4 (0.40) KCNN4KIF11MAPK1ALDH1A1
SCHEMBL8945088 0.73 KCNN4 (0.40) KCNN4KIF11MAPK1ALDH1A1
SCHEMBL3302423 0.72 KCNN4 (0.47) KCNN4MAPTKIF11KDM4ELMNA
SCHEMBL3302429 0.72 KCNN4 (0.47) KCNN4MAPTKIF11KDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6448261-B1 CORTICOTROPIN RELEASING FACTOR ANTAGONISTS; TREATING ANXIETY, DEPRESSION, AND OTHER PSYCHIATRIC AND NEUROLOGICAL DISORDERS BRISTOL-MYERS SQUIBB PHARMA COMPANY 2002-09-10 US disclosed
EP-0935601-A4 ARYLAMINO FUSED PYRIDINES AND PYRIMIDINES DU PONT PHARM CO (US) 2002-08-07 EP disclosed
US-6107300-A CORTICOTROPIN RELEASING FACTOR ANTAGONIST; PSYCHOLOGICAL DISORDERS DUPONT PHARMACEUTICALS (US) 2000-08-22 US disclosed
EP-0935601-A2 ARYLAMINO FUSED PYRIDINES AND PYRIMIDINES Du Pont Pharmaceuticals Company (US) 1999-08-18 EP disclosed
WO-1997035539-A2 ARYLAMINO FUSED PYRIDINES AND PYRIMIDINES DU PONT PHARMACEUTICALS COMPANY (US) 1997-10-02 WO disclosed