SCHEMBL7486456

SCHEMBL7486456

CCN1CCC2(c3cccc(OC)c3)CC(=O)CCC2C1

nearest known ligand 0.60

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 4/20 0.60
OPRD1 P41143 4/20 0.60
OPRK1 P41145 4/20 0.60
SLC6A4 P31645 2/20 0.48
SLC6A2 P23975 1/20 0.47
SLC6A3 Q01959 1/20 0.47
SIGMAR1 Q99720 2/20 0.45
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
CXCR3 P49682 1/20 0.42
CTSD P07339 1/20 0.41
CTSE P14091 1/20 0.41
BACE1 P56817 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7486453 1.00 OPRM1 (0.60) OPRM1OPRD1OPRK1SLC6A4SLC6A2
Hydrochloric Acid SCHEMBL7487249 0.99 OPRM1 (0.59) OPRM1OPRD1OPRK1SLC6A4SLC6A2
Hydrochloric Acid SCHEMBL7487248 0.99 OPRM1 (0.59) OPRM1OPRD1OPRK1SLC6A4SLC6A2
SCHEMBL7482382 0.90 OPRM1 (0.56) OPRM1OPRD1OPRK1SLC6A4SLC6A2
SCHEMBL7482389 0.90 OPRM1 (0.56) OPRM1OPRD1OPRK1SLC6A4SLC6A2
SCHEMBL11398571 0.89 OPRD1 (0.76) OPRM1OPRD1OPRK1SLC6A4SLC6A2
SCHEMBL8396855 0.89 OPRD1 (0.76) OPRM1OPRD1OPRK1SLC6A4SLC6A2
SCHEMBL8396856 0.89 OPRD1 (0.76) OPRM1OPRD1OPRK1SLC6A4SLC6A2
Hydrochloric Acid SCHEMBL7496002 0.89 OPRM1 (0.56) OPRM1OPRD1OPRK1SLC6A4SLC6A2
Hydrochloric Acid SCHEMBL7496005 0.89 OPRM1 (0.56) OPRM1OPRD1OPRK1SLC6A4SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0712402-B1 HYDROISOQUINOLINE DERIVATIVES SMITHKLINE BEECHAM SPA (IT) 2002-04-10 EP disclosed
EP-0854868-A1 SUBSTITUTED HYDROISOQUINOLINE DERIVATIVES AND THEIR USE AS PHARMACEUTICALS Smithkline Beecham S.p.A. (IT) 1998-07-29 EP disclosed
WO-1997010216-A1 SUBSTITUTED HYDROISOQUINOLINE DERIVATIVES AND THEIR USE AS PHARMACEUTICALS SMITHKLINE BEECHAM S.P.A. (IT) 1997-03-20 WO disclosed