SCHEMBL748784

SCHEMBL748784

O[C@H]1CNCC[C@H]1N(Cc1ccccc1)Cc1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 5/20 0.49
SLC6A4 P31645 5/20 0.49
GBA1 P04062 2/20 0.47
SLC18A3 Q16572 3/20 0.45
CTSD P07339 1/20 0.43
SLC6A3 Q01959 4/20 0.42
EBP Q15125 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16422495 0.85 CTSD (0.54) SLC6A2SLC6A4GBA1SLC18A3CTSD
SCHEMBL9531212 0.84 SLC18A3 (0.66) SLC6A2SLC6A4GBA1SLC18A3CTSD
SCHEMBL2776534 0.84 CTSD (0.55) SLC6A2SLC6A4GBA1SLC18A3CTSD
SCHEMBL9531228 0.84 SLC18A3 (0.66) SLC6A2SLC6A4GBA1SLC18A3CTSD
SCHEMBL2776529 0.84 CTSD (0.55) SLC6A2SLC6A4GBA1SLC18A3CTSD
SCHEMBL9531221 0.84 SLC18A3 (0.66) SLC6A2SLC6A4GBA1SLC18A3CTSD
SCHEMBL8245028 0.83 SLC6A2 (0.51) SLC6A2SLC6A4GBA1SLC18A3CTSD
SCHEMBL22273230 0.81 SLC18A3 (0.56) SLC6A2SLC6A4SLC18A3CTSDEBP
SCHEMBL22252483 0.81 SLC18A3 (0.56) SLC6A2SLC6A4SLC18A3CTSDEBP
SCHEMBL20687903 0.81 SLC18A3 (0.56) SLC6A2SLC6A4SLC18A3CTSDEBP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138204-B2 Emesis, dyspepsia, gastroparesis, constipation, gastroesophageal reflux, or post-operative ileus; cisapride analogs; side effect reduction of adverse events; (R)-quinuclidin-3-yl 6-((3S,4R)-4-(4-amino-5-chloro-2-methoxybenzamido)-3-methoxypiperidin-1-yl)hexanoate or salts ARYX THERAPEUTICS, INC. (US) 2012-03-20 US disclosed
US-7326787-B2 Synthetic methods and intermediates for stereoisomeric compounds useful for the treatment of gastrointestinal and central nervous system disorders ARYX THERAPEUTICS, INC. (US) 2008-02-05 US disclosed