SCHEMBL7488589

SCHEMBL7488589

CCOC(=O)Cn1c(=O)c(=O)[nH]c2ccc3ccc(N)cc3c21

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 2/20 0.44
GRIA1 P42261 2/20 0.41
GRIA2 P42262 2/20 0.41
GRIA3 P42263 2/20 0.41
GRIA4 P48058 2/20 0.41
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
TDP1 Q9NUW8 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
TNF P01375 2/20 0.40
TSHR P16473 2/20 0.40
CYP1A2 P05177 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
KDM4E B2RXH2 3/20 0.39
RAB9A P51151 2/20 0.39
ALDH1A1 P00352 4/20 0.39
MAPK1 P28482 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.37
GAA P10253 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7481432 0.89 TNF (0.45) ADORA3TNFKDM4EALDH1A1HSD17B10
SCHEMBL7486654 0.85 CYP1A2 (0.49) MEN1KMT2ATDP1L3MBTL1TNF
SCHEMBL8608979 0.84 TSHR (0.40) GRIA1GRIA2GRIA3GRIA4MEN1
SCHEMBL7477922 0.84 ADORA3 (0.52) ADORA3GRIA1GRIA2GRIA3GRIA4
SCHEMBL7477314 0.83 GRIA1 (0.48) GRIA1GRIA2GRIA3GRIA4MEN1
SCHEMBL8609389 0.83 ALDH1A1 (0.41) ADORA3GRIA1GRIA2GRIA3GRIA4
SCHEMBL8674575 0.79 GRIA1 (0.43) ADORA3GRIA1GRIA2GRIA3GRIA4
SCHEMBL7656452 0.79 GRIA1 (0.57) ADORA3GRIA1GRIA2GRIA3GRIA4
SCHEMBL7484293 0.75 TNF (0.50) KMT2ATDP1TNFKDM4EALDH1A1
SCHEMBL7475364 0.74 GRIK1 (0.53) GRIA1GRIA2GRIA3GRIA4MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0799224-B1 QUINOXALINES AND DRUGS PREPARED THEREFROM BASF AG (DE) 2002-04-17 EP disclosed
US-5849743-A Quinoxalines and drugs prepared therefrom BASF AKTIENGESELLSCHAFT (DE) 1998-12-15 US disclosed
EP-0760811-A1 IMIDAZOLE DERIVATIVES AS HISTAMINE RECEPTOR H 3? (ANT)AGONISTS INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 1997-03-12 EP disclosed
WO-1996019476-A1 NOVEL QUINOXALINES AND DRUGS PREPARED THEREFROM BASF AKTIENGESELLSCHAFT (DE) 1996-06-27 WO disclosed
EP-0572852-A1 Quinoxalin-2,3(1H,4H)-diones used as medicine BASF Aktiengesellschaft (DE) 1993-12-08 EP disclosed