SCHEMBL7488974

SCHEMBL7488974

Cc1oc(-c2ccccc2)nc1CCC(O)c1ccc(CC2NC(=O)OC2=O)cc1

nearest known ligand 0.45

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PPARG P37231 19/20 0.45
PPARA Q07869 15/20 0.44
KDM4E B2RXH2 1/20 0.41
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
KCNH2 Q12809 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7494345 0.92 PPARG (0.47) PPARGPPARAKDM4E
SCHEMBL7486254 0.90 PPARG (0.49) PPARGPPARA
SCHEMBL7487592 0.84 PPARG (0.47) PPARGPPARACYP3A4CYP2C9KCNH2
SCHEMBL7909696 0.83 PPARG (0.60) PPARGPPARACYP3A4CYP2C9KCNH2
SCHEMBL9274342 0.80 PPARG (0.47) PPARGPPARACYP3A4CYP2C9KCNH2
SCHEMBL7877637 0.80 PPARG (0.47) PPARGPPARACYP3A4CYP2C9KCNH2
SCHEMBL9286066 0.80 PPARG (0.47) PPARGPPARACYP3A4CYP2C9KCNH2
SCHEMBL7877640 0.80 PPARG (0.47) PPARGPPARACYP3A4CYP2C9KCNH2
SCHEMBL7879128 0.80 PPARG (0.47) PPARGPPARACYP3A4CYP2C9KCNH2
SCHEMBL7494333 0.79 PPARG (0.47) PPARGPPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0643050-B1 Oxazolidinedione derivatives and their use as hypoglycemic agent TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2002-04-10 EP claimed
EP-0643050-A1 Oxazolidinedione derivatives and their use as hypoglycemic agent Takeda Chemical Industries, Ltd. (JP) 1995-03-15 EP claimed
US-5614544-A HYPOGLYCEMIC AND HYPOLIPIDEMIC AGENTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-03-25 US disclosed
EP-0643050-A1 Oxazolidinedione derivatives and their use as hypoglycemic agent Takeda Chemical Industries, Ltd. (JP) 1995-03-15 EP disclosed