SCHEMBL7489293

SCHEMBL7489293

O=C(Nc1ccc([N+](=O)[O-])cc1O)Nc1ccccc1F.O=C(Nc1ccc([N+](=O)[O-])cc1O)Nc1ccccc1[N+](=O)[O-]

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 8/20 0.67
KMT2A Q03164 8/20 0.67
MAPT P10636 6/20 0.67
HTT P42858 4/20 0.67
RAB9A P51151 3/20 0.67
LMNA P02545 3/20 0.67
NPC1 O15118 2/20 0.67
MAPK1 P28482 1/20 0.67
CXCR1 P25024 3/20 0.65
CXCR2 P25025 3/20 0.65
TDP1 Q9NUW8 1/20 0.65
HDAC6 Q9UBN7 1/20 0.65
KCNMA1 Q12791 3/20 0.57
CA12 O43570 2/20 0.53
CA1 P00915 2/20 0.53
CA9 Q16790 2/20 0.53
RORC P51449 1/20 0.53
SMN1; SMN2 Q16637 3/20 0.51
ALDH1A1 P00352 1/20 0.51
NPSR1 Q6W5P4 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5595038 0.94 MEN1 (0.74) MEN1KMT2AMAPTHTTRAB9A
SCHEMBL5595118 0.93 CXCR2 (0.74) MEN1KMT2AMAPTHTTRAB9A
SCHEMBL5595106 0.83 KMT2A (0.69) MEN1KMT2AMAPTHTTRAB9A
SCHEMBL6920109 0.83 CXCR1 (0.66) MEN1KMT2AMAPTHTTRAB9A
SCHEMBL5594659 0.83 CXCR1 (0.66) MEN1KMT2AMAPTHTTRAB9A
SCHEMBL7489294 0.82 KMT2A (0.51) MEN1KMT2AMAPTHTTRAB9A
SCHEMBL5595104 0.82 CXCR1 (0.80) MEN1KMT2AMAPTHTTRAB9A
SCHEMBL6824010 0.81 KMT2A (0.50) MEN1KMT2AMAPTHTTRAB9A
SCHEMBL7494939 0.80 CXCR2 (0.63) MEN1KMT2AMAPTHTTRAB9A
SCHEMBL3706835 0.80 KMT2A (0.74) MEN1KMT2AMAPTHTTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0896531-A4 IL-8 RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 2002-10-30 EP disclosed
EP-0896531-A1 IL-8 RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1999-02-17 EP disclosed
WO-1997029743-A1 IL-8 RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1997-08-21 WO disclosed