SCHEMBL7494073

SCHEMBL7494073

c1ccc(Cc2cc(C3CCNCC3)on2)cc1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.49
RAB9A P51151 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
TDP1 Q9NUW8 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.49
SLC6A3 Q01959 1/20 0.45
GABRA1 P14867 2/20 0.44
GABRB2 P47870 1/20 0.44
HTR2C P28335 1/20 0.43
HTR2B P41595 1/20 0.43
BCHE P06276 1/20 0.43
ACHE P22303 1/20 0.43
GABRG2 P18507 1/20 0.43
GABRB3 P28472 1/20 0.43
PLAT P00750 1/20 0.43
GBA1 P04062 1/20 0.42
S1PR1 P21453 1/20 0.42
S1PR3 Q99500 1/20 0.42
HRH1 P35367 1/20 0.42
SLC18A3 Q16572 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL7502182 0.89 S1PR3 (0.43) ALDH1A1RAB9ASMN1; SMN2TDP1L3MBTL1
SCHEMBL8105457 0.77 ALDH1A1 (0.47) ALDH1A1RAB9ASMN1; SMN2TDP1L3MBTL1
SCHEMBL2210707 0.77 NPC1 (0.63) RAB9ASLC6A3BCHEACHEPLAT
SCHEMBL7505745 0.75 GABRA1 (0.46) SLC6A3GABRA1GABRB2GABRG2GABRB3
SCHEMBL5765171 0.75 USP7 (0.47) SLC6A3GABRA1GABRB2HTR2BBCHE
SCHEMBL3120592 0.74 SMYD3 (0.43) GABRA1BCHEACHEGABRG2GABRB3
SCHEMBL5764334 0.73 MKNK1 (0.47) GABRA1GABRB2HTR2CHTR2BGABRG2
SCHEMBL3868513 0.72 NMT1 (0.55) PLATNMT1
Hydrochloric Acid SCHEMBL5765492 0.72 GABRA1 (0.46) GABRA1GABRB2HTR2CHTR2BGABRG2
Hydrochloric Acid SCHEMBL3597129 0.71 NMT1 (0.54) GABRA1GABRB2PLATNMT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1171122-A4 PYRROLIDINE MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY MERCK & CO INC (US) 2002-05-29 EP disclosed
EP-1171122-A1 PYRROLIDINE MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY Merck & Co., Inc. (US) 2002-01-16 EP disclosed
US-6248755-B1 ANTIINFLAMMATORY AGENTS; ANTIALLERGENS; AUTOIMMUNE DISEASES MERCK & CO., INC. 2001-06-19 US disclosed
WO-2000059502-A1 PYRROLIDINE MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY MERCK & CO., INC. (US) 2000-10-12 WO disclosed