SCHEMBL7494202

SCHEMBL7494202

CCOC(=O)CC(=O)C=NNc1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 8/20 0.49
ALDH1A1 P00352 6/20 0.49
MAPT P10636 6/20 0.49
RAB9A P51151 5/20 0.49
KMT2A Q03164 3/20 0.49
MAPK1 P28482 1/20 0.49
PRNP P04156 1/20 0.47
ALOX12 P18054 1/20 0.47
LMNA P02545 4/20 0.46
NPC1 O15118 4/20 0.45
SMN1; SMN2 Q16637 3/20 0.45
HPGD P15428 1/20 0.45
ATM Q13315 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.44
TDP1 Q9NUW8 2/20 0.43
NOX1 Q9Y5S8 2/20 0.43
MEN1 O00255 2/20 0.43
HTT P42858 1/20 0.42
GLA P06280 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27332500 0.85 ALDH1A1 (0.44) GAAALDH1A1MAPTRAB9AKMT2A
SCHEMBL14059066 0.83 MAPT (0.52) GAAALDH1A1MAPTRAB9AKMT2A
SCHEMBL14269202 0.83 MAPT (0.52) GAAALDH1A1MAPTRAB9AKMT2A
SCHEMBL14059065 0.83 MAPT (0.52) GAAALDH1A1MAPTRAB9AKMT2A
SCHEMBL10027943 0.82 NOX1 (0.47) GAAALDH1A1MAPTRAB9AKMT2A
SCHEMBL23728219 0.80 NOX1 (0.49) GAAALDH1A1MAPTRAB9AKMT2A
SCHEMBL23728221 0.80 NOX1 (0.49) GAAALDH1A1MAPTRAB9AKMT2A
SCHEMBL7490760 0.79 MAPT (0.48) GAAALDH1A1MAPTRAB9AKMT2A
SCHEMBL5817859 0.76 MAPT (0.49) GAAALDH1A1MAPTRAB9AKMT2A
SCHEMBL9974840 0.76 ALDH1A1 (0.58) GAAALDH1A1MAPTRAB9AKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0712402-B1 HYDROISOQUINOLINE DERIVATIVES SMITHKLINE BEECHAM SPA (IT) 2002-04-10 EP disclosed
US-5731322-A ADMINISTERING AS ANALGESICS OR IMMUNOMODULATING AND/OR CARDIOVASCULAR AGENTS SMITHKLINE BEECHAM S.P.A. (IT) 1998-03-24 US disclosed
EP-0712402-A1 HYDROISOQUINOLINE DERIVATIVES Smithkline Beecham S.p.A. (IT) 1996-05-22 EP disclosed
WO-1995004734-A1 HYDROISOQUINOLINE DERIVATIVES SMITHKLINE BEECHAM FARMACEUTICI S.P.A. (IT) 1995-02-16 WO disclosed