SCHEMBL7494472

SCHEMBL7494472

COc1c(N2CC3CCOC3(CNC(=O)OC(C)(C)C)C2)c(F)c(N)c2c(=O)c(OC(=O)O)cn(C3CC3)c12

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 7/20 0.36
KCNH2 Q12809 4/20 0.35
POLB P06746 3/20 0.35
CACNA1F O60840 1/20 0.35
MAPK1 P28482 1/20 0.35
CACNA1D Q01668 1/20 0.35
CACNA1S Q13698 1/20 0.35
CACNA1C Q13936 1/20 0.35
KDM4E B2RXH2 4/20 0.31
ALDH1A1 P00352 3/20 0.31
TDP1 Q9NUW8 2/20 0.31
HPGD P15428 2/20 0.31
PRKD3 O94806 1/20 0.31
ALOX15 P16050 1/20 0.31
OPRM1 P35372 1/20 0.31
CLK2 P49760 1/20 0.31
HSD17B10 Q99714 1/20 0.31
CLK4 Q9HAZ1 1/20 0.31
LMNA P02545 2/20 0.31
NPSR1 Q6W5P4 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9212277 0.94 CACNA1F (0.40) GSK3BKCNH2POLBCACNA1FMAPK1
SCHEMBL7494469 0.91 GSK3B (0.46) GSK3BKCNH2POLBCACNA1FMAPK1
SCHEMBL9207351 0.88 MEN1 (0.39) KCNH2POLBCACNA1FMAPK1CACNA1D
SCHEMBL7546072 0.88 KCNH2 (0.39) GSK3BKCNH2POLBCACNA1FMAPK1
Hydrochloric Acid SCHEMBL7491976 0.87 KCNH2 (0.39) GSK3BKCNH2POLBCACNA1FMAPK1
SCHEMBL7493085 0.87 KCNH2 (0.45) GSK3BKCNH2POLBKDM4EALDH1A1
Trifluoroacetic Acid SCHEMBL7499704 0.86 KCNH2 (0.37) GSK3BKCNH2POLBCACNA1FMAPK1
SCHEMBL8924239 0.85 CACNA1F (0.52) GSK3BKCNH2POLBCACNA1FMAPK1
SCHEMBL9228860 0.84 MEN1 (0.32) KCNH2POLBCACNA1FMAPK1CACNA1D
SCHEMBL7496654 0.84 KCNH2 (0.37) KCNH2POLBKDM4EALDH1A1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0944385-B1 USE OF 7-(1-AMINOMETHYL-2-OXA-7-AZA-BICYCLO 3.3.0]OCT-7-YL)-QUINOLONE CARBOXYLIC ACID AND NAPHTHYRIDONE CARBOXYLIC ACID DERIVATIVES FOR TREATING HELICOBACTER PYLORI INFECTIONS AND THE GASTRODUODENAL DISEASES ASSOCIATED THEREWITH BAYER AG (DE) 2002-10-16 EP disclosed