SCHEMBL7497232

SCHEMBL7497232

Nc1nc(O)c2c(n1)NCC(CCc1cc(C(=O)N[C@@H](CCC(=O)O)C(=O)O)ns1)C2

nearest known ligand 0.60

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
GART P22102 12/20 0.52
DHFR P00374 3/20 0.46
FOLR1 P15328 2/20 0.40
ATIC P31939 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7502144 0.93 GART (0.53) GARTDHFRFOLR1
SCHEMBL7498884 0.87 GART (0.53) GARTDHFRFOLR1ATIC
SCHEMBL9383090 0.86 GART (0.56) GARTDHFRFOLR1ATIC
SCHEMBL14403392 0.86 DHFR (0.59) GARTDHFRFOLR1ATIC
SCHEMBL9383067 0.86 DHFR (0.59) GARTDHFRFOLR1ATIC
SCHEMBL9381796 0.86 DHFR (0.59) GARTDHFRFOLR1ATIC
SCHEMBL8018583 0.86 GART (0.54) GARTDHFRFOLR1ATIC
SCHEMBL7499714 0.86 GART (0.54) GARTDHFRFOLR1ATIC
SCHEMBL9380609 0.86 DHFR (0.59) GARTDHFRFOLR1ATIC
SCHEMBL9381786 0.86 DHFR (0.59) GARTDHFRFOLR1ATIC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0904271-A4 5,6,7,8-TETRAHYDROPYRIDO[2,3-d]PYRIMIDINES UNIV PRINCETON (US) 2002-01-23 EP disclosed
US-6066639-A ANTITUMOR AGENTS THE TRUSTEES OF PRINCETON UNIVERSITY (US) 2000-05-23 US disclosed
EP-0904271-A1 5,6,7,8-TETRAHYDROPYRIDO[2,3-d]PYRIMIDINES THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1999-03-31 EP disclosed
WO-1997041115-A1 5,6,7,8-TETRAHYDROPYRIDO[2,3-d]PYRIMIDINES THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1997-11-06 WO disclosed