SCHEMBL7497451

SCHEMBL7497451

COC(=O)CC[C@H](NC(=O)c1ccc(CCC2CNc3nc(N)nc(O)c3C2)[nH]1)C(=O)OC

nearest known ligand 0.48

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GART P22102 6/20 0.43
DHFR P00374 3/20 0.39
ATIC P31939 3/20 0.33
CA12 O43570 1/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
CA9 Q16790 1/20 0.32
ALDH1A1 P00352 1/20 0.31
MAPK1 P28482 1/20 0.31
ALOX5 P09917 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7497455 1.00 GART (0.43) GARTDHFRATICCA12CA1
SCHEMBL7553633 0.87 GART (0.58) GARTDHFRATIC
SCHEMBL7496781 0.87 GART (0.58) GARTDHFRATIC
SCHEMBL8017846 0.86 GART (0.40) GARTDHFRCA12CA1CA2
SCHEMBL8017849 0.86 GART (0.40) GARTDHFRCA12CA1CA2
SCHEMBL7496547 0.85 GART (0.43) GARTDHFRATICALOX5
SCHEMBL7497802 0.85 GART (0.43) GARTDHFRATICALDH1A1MAPK1
SCHEMBL7496744 0.79 GART (0.58) GARTDHFRATIC
SCHEMBL7494746 0.79 DHFR (0.42) GARTDHFR
SCHEMBL9383614 0.77 GART (0.56) GARTDHFRATICALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0904271-A4 5,6,7,8-TETRAHYDROPYRIDO[2,3-d]PYRIMIDINES UNIV PRINCETON (US) 2002-01-23 EP disclosed
US-6066639-A ANTITUMOR AGENTS THE TRUSTEES OF PRINCETON UNIVERSITY (US) 2000-05-23 US disclosed
EP-0904271-A1 5,6,7,8-TETRAHYDROPYRIDO[2,3-d]PYRIMIDINES THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1999-03-31 EP disclosed
WO-1997041115-A1 5,6,7,8-TETRAHYDROPYRIDO[2,3-d]PYRIMIDINES THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1997-11-06 WO disclosed